SCHEMBL8535454

SCHEMBL8535454

N#Cc1cccc(CN(CCN2CCN(Cc3cccc(C(F)(F)F)c3)CC2)C2CCCCCC2)c1

nearest known ligand 0.50

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.50
ALDH1A1 P00352 1/20 0.50
GAA P10253 1/20 0.50
TACR1 P25103 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.43
LMNA P02545 1/20 0.42
SLC6A2 P23975 2/20 0.42
SLC6A4 P31645 2/20 0.42
SLC6A3 Q01959 1/20 0.42
CLPP Q16740 1/20 0.42
HRH3 Q9Y5N1 3/20 0.40
SIGMAR1 Q99720 1/20 0.40
HTR1A P08908 1/20 0.40
CYP3A4 P08684 1/20 0.40
KCNH2 Q12809 1/20 0.40
CHIT1 Q13231 1/20 0.40
CHIA Q9BZP6 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8539056 1.00 KDM4E (0.50) KDM4EALDH1A1GAATACR1L3MBTL1
SCHEMBL8540937 0.92 SLC6A2 (0.47) SLC6A2SLC6A4SLC6A3HRH3KCNH2
SCHEMBL8535362 0.91 KDM4E (0.60) KDM4EALDH1A1GAALMNASLC6A2
SCHEMBL8542233 0.89 SLC6A2 (0.43) TACR1SLC6A2SLC6A4SLC6A3HRH3
SCHEMBL8535949 0.88 SLC6A2 (0.46) SLC6A2SLC6A4SLC6A3HRH3
SCHEMBL8542251 0.87 KDM4E (0.54) KDM4EALDH1A1GAALMNASLC6A2
SCHEMBL8537719 0.87 SLC6A2 (0.45) KDM4EALDH1A1SLC6A2SLC6A4SLC6A3
SCHEMBL8541455 0.87 KDM4E (0.54) KDM4EALDH1A1GAALMNASLC6A2
SCHEMBL8536918 0.86 ALDH1A1 (0.53) KDM4EALDH1A1GAALMNASLC6A2
SCHEMBL8588892 0.83 RORC (0.48) KDM4EALDH1A1L3MBTL1SLC6A2SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5817489-A BACTERICIDES, OR CHEMICAL INTERMEDIATES THEREOF; DRUG LIBRARIES ISIS PHARMACEUTICALS, INC. (US) 1998-10-06 US claimed