SCHEMBL8535718

SCHEMBL8535718

COCC1(COC)Oc2ccc(Br)cc2[C@@H]2O[C@@H]21

nearest known ligand 0.34

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 4/20 0.34
HTR2C P28335 4/20 0.34
DRD2 P14416 2/20 0.34
ADRA2A P08913 1/20 0.34
ADRA2C P18825 1/20 0.34
DRD1 P21728 1/20 0.34
HTR7 P34969 1/20 0.34
HRH1 P35367 1/20 0.34
DRD3 P35462 1/20 0.34
IDO1 P14902 2/20 0.32
HTR2B P41595 5/20 0.32
AHR P35869 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8540483 0.86 HTR2A (0.33) HTR2AHTR2CDRD2ADRA2AADRA2C
SCHEMBL9735917 0.85 HTR2A (0.39) HTR2AHTR2CDRD2ADRA2AADRA2C
SCHEMBL8537452 0.83 TRPV1 (0.35) HTR2AHTR2CDRD2ADRA2AADRA2C
SCHEMBL8534906 0.80 ABCB1 (0.41)
SCHEMBL8535501 0.80 ABCB1 (0.41)
SCHEMBL8534900 0.80 ABCB1 (0.41)
SCHEMBL8536317 0.78 MAPT (0.39)
SCHEMBL4848406 0.77 HTR2A (0.32) HTR2AHTR2CDRD2ADRA2AADRA2C
SCHEMBL4020277 0.77 HTR2A (0.32) HTR2AHTR2CDRD2ADRA2AADRA2C
SCHEMBL9141916 0.76 HTR2A (0.36) HTR2AHTR2CDRD2ADRA2AADRA2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5719155-A CARDIOVASCULAR DISORDERS JAPAN TOBACCO INC. (JP) 1998-02-17 US disclosed
EP-0677519-A1 CHROMAN DERIVATIVE AND MEDICINAL USE THEREOF Japan Tobacco Inc. (JP) 1995-10-18 EP disclosed