SCHEMBL8536130

SCHEMBL8536130

NN=CNc1cccc(S(=O)(=O)C(N)(Cc2c(F)c(F)c(-c3ccccc3)c(F)c2F)C(=O)O)c1

nearest known ligand 0.35

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CA1 P00915 12/20 0.35
CA2 P00918 12/20 0.35
CA4 P22748 3/20 0.35
HSD17B1 P14061 3/20 0.35
HSD17B2 P37059 3/20 0.35
CA9 Q16790 7/20 0.34
CA12 O43570 6/20 0.34
MAPT P10636 1/20 0.33
F2 P00734 1/20 0.32
TMPRSS6 Q8IU80 1/20 0.32
SLC1A3 P43003 1/20 0.32
SLC1A2 P43004 1/20 0.32
SLC1A1 P43005 1/20 0.32
ITGB3 P05106 1/20 0.31
ITGB1 P05556 1/20 0.31
ITGAV P06756 1/20 0.31
ITGA2B P08514 1/20 0.31
ITGA5 P08648 1/20 0.31
ITGB5 P18084 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8499997 0.74 PFKFB3 (0.41) CA1CA2HSD17B1HSD17B2MAPT
SCHEMBL8697026 0.72 CA1 (0.40) CA1CA2CA4CA9CA12
SCHEMBL8532207 0.72 CA1 (0.33) CA1CA2CA4CA9CA12
SCHEMBL8531518 0.70 CA1 (0.34) CA1CA2CA4CA9CA12
SCHEMBL8536202 0.69 FFAR1 (0.35) CA1CA2CA4CA9CA12
SCHEMBL8429166 0.68 CA1 (0.43) CA1CA2CA4HSD17B1HSD17B2
SCHEMBL8501213 0.64 CA12 (0.40) CA1CA2CA9CA12ITGB3
SCHEMBL8693780 0.64 CA1 (0.39) CA1CA2CA4HSD17B1HSD17B2
SCHEMBL8499992 0.64 MEN1 (0.42) CA1CA2HSD17B1HSD17B2MAPT
SCHEMBL8694027 0.63 CA1 (0.38) CA1CA2CA4HSD17B1HSD17B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5773646-A INTEGRIN INHIBITORS G. D. SEARLE & CO. (US) 1998-06-30 US disclosed