SCHEMBL8536671

SCHEMBL8536671

COc1ccc(CSC)c(-c2ncc[nH]2)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 1/20 0.46
NOS1 P29475 1/20 0.46
NOS2 P35228 1/20 0.46
ADRA2A P08913 1/20 0.40
ADRA2C P18825 1/20 0.40
ADRA1D P25100 1/20 0.40
ADRA1A P35348 1/20 0.40
ADRA1B P35368 1/20 0.40
CYP19A1 P11511 2/20 0.40
CYP1A2 P05177 2/20 0.40
CYP3A4 P08684 2/20 0.40
CYP2D6 P10635 2/20 0.40
CYP2C9 P11712 2/20 0.40
CYP2C19 P33261 2/20 0.40
MC4R P32245 2/20 0.39
TLK2 Q86UE8 2/20 0.39
SMPD3 Q9NY59 1/20 0.38
ALDH1A1 P00352 2/20 0.36
GRK6 P43250 2/20 0.36
MEN1 O00255 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8539649 0.90 NOS3 (0.47) NOS3NOS1NOS2ADRA2AADRA2C
SCHEMBL7460509 0.83 MC4R (0.43) ADRA2AADRA2CADRA1DADRA1AADRA1B
SCHEMBL8537559 0.82 MC4R (0.44) ADRA2AADRA2CCYP19A1CYP1A2CYP3A4
SCHEMBL8541205 0.82 NISCH (0.36) ADRA2AADRA2CADRA1ACYP19A1CYP1A2
SCHEMBL8541277 0.81 JAK2 (0.44) ADRA1ACYP19A1CYP1A2CYP3A4CYP2D6
SCHEMBL8543161 0.81 SMPD3 (0.46) NOS3NOS1NOS2ADRA1ACYP19A1
SCHEMBL31429681 0.77 NOTUM (0.53) ADRA2AADRA2CADRA1DADRA1AADRA1B
SCHEMBL31559158 0.77 SMPD3 (0.50) ADRA2AADRA2CADRA1DADRA1AADRA1B
SCHEMBL8537087 0.77 CSNK1A1 (0.45) ADRA2AADRA2CADRA1ACYP19A1CYP1A2
SCHEMBL8541036 0.77 SMPD3 (0.50) ADRA2AADRA2CADRA1DADRA1AADRA1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0857171-A2 IMIDAZOLE DERIVATIVES AND THE USE THEREOF AS NITROGEN MONOXIDE SYNTHASE INHIBITORS SCHERING AKTIENGESELLSCHAFT (DE) 1998-08-12 EP disclosed
WO-1997015555-A2 IMIDAZOLE DERIVATIVES AND THE USE THEREOF AS NITROGEN MONOXIDE SYNTHASE INHIBITORS SCHERING AKTIENGESELLSCHAFT (DE) 1997-05-01 WO disclosed