SCHEMBL8543161

SCHEMBL8543161

COc1cc(CSC)c(-c2ncc[nH]2)cc1OC

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMPD3 Q9NY59 1/20 0.46
MC4R P32245 2/20 0.43
P2RX3 P56373 1/20 0.39
P2RX2 Q9UBL9 1/20 0.39
TLK2 Q86UE8 1/20 0.37
CDK4 P11802 1/20 0.37
CCNA2 P20248 1/20 0.37
CCND1 P24385 1/20 0.37
CDK2 P24941 1/20 0.37
CCND3 P30281 1/20 0.37
TUBB4A P04350 1/20 0.36
TUBB P07437 1/20 0.36
TUBA3C P0DPH7 1/20 0.36
TUBA1B P68363 1/20 0.36
TUBA4A P68366 1/20 0.36
TUBB4B P68371 1/20 0.36
TUBB3 Q13509 1/20 0.36
TUBB2A Q13885 1/20 0.36
TUBB8 Q3ZCM7 1/20 0.36
TUBA3E Q6PEY2 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8539649 0.82 NOS3 (0.47) SMPD3MC4RTLK2CDK4CCNA2
SCHEMBL8536671 0.81 NOS3 (0.46) SMPD3MC4RTLK2NOS3NOS1
SCHEMBL8540730 0.78 MC4R (0.46) SMPD3MC4RALDH1A1CYP1A2CYP3A4
SCHEMBL8540790 0.77 NISCH (0.37) SMPD3MC4RNOS3NOS1NOS2
SCHEMBL8541205 0.75 NISCH (0.36) SMPD3MC4RALDH1A1CYP1A2CYP3A4
SCHEMBL8541400 0.75 MC4R (0.37) MC4RALDH1A1CYP1A2CYP3A4CYP2D6
SCHEMBL8537559 0.75 MC4R (0.44) SMPD3MC4RALDH1A1CYP1A2CYP3A4
SCHEMBL8536816 0.75 JAK2 (0.47) SMPD3MC4RCDK4CCNA2CCND1
SCHEMBL8540597 0.75 CSNK1A1 (0.36) SMPD3MC4RP2RX3P2RX2ALDH1A1
SCHEMBL8541277 0.74 JAK2 (0.44) SMPD3MC4RCDK4CCNA2CCND1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0857171-A2 IMIDAZOLE DERIVATIVES AND THE USE THEREOF AS NITROGEN MONOXIDE SYNTHASE INHIBITORS SCHERING AKTIENGESELLSCHAFT (DE) 1998-08-12 EP disclosed
WO-1997015555-A2 IMIDAZOLE DERIVATIVES AND THE USE THEREOF AS NITROGEN MONOXIDE SYNTHASE INHIBITORS SCHERING AKTIENGESELLSCHAFT (DE) 1997-05-01 WO disclosed