SCHEMBL8537191

SCHEMBL8537191

CC(C)(C)[Si](Oc1cccc(C#N)c1)(c1ccccc1)c1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 1/20 0.42
GABRA1 P14867 1/20 0.38
GABRG2 P18507 1/20 0.38
GABRB3 P28472 1/20 0.38
GABRA5 P31644 1/20 0.38
GABRA3 P34903 1/20 0.38
TSHR P16473 1/20 0.37
SLC6A2 P23975 2/20 0.36
SLC6A4 P31645 2/20 0.36
FFAR1 O14842 1/20 0.36
SLC6A3 Q01959 1/20 0.36
PGR P06401 1/20 0.36
TBXAS1 P24557 1/20 0.36
MGLL Q99685 1/20 0.35
VEGFA P15692 1/20 0.35
EPAS1 Q99814 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
ACP1 P24666 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28574194 0.85 FABP7 (0.40) BACE1
SCHEMBL8002249 0.81 HAO1 (0.44)
SCHEMBL704145 0.79 CA4 (0.37) TSHRSMN1; SMN2
SCHEMBL7092637 0.78 CYP3A4 (0.42) TSHR
SCHEMBL3287158 0.78 CA12 (0.41) SLC6A2SLC6A4SLC6A3TBXAS1MGLL
SCHEMBL7227692 0.78 HAO1 (0.40) BACE1GABRA1GABRG2GABRB3GABRA5
SCHEMBL4470099 0.77 MAOB (0.42) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL31637439 0.77 MAOB (0.49) TSHR
SCHEMBL8135354 0.77
SCHEMBL29910455 0.77 MAOB (0.42) GABRA1GABRG2GABRB3GABRA5GABRA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5770598-A ANTITUMOR AGENTS; REACTING WITH CARBONYL DIIMIDAZOLE AND AMIDOXIMES UNIVERSITY COLLEGE CARDIFF CONSULTANTS LIMITED (GB) 1998-06-23 US disclosed
EP-0769012-A1 TETRACYCLIC DERIVATIVES AND THEIR USE AS ANTITUMOUR AGENTS THE WELLCOME FOUNDATION LIMITED (GB) 1997-04-23 EP disclosed
WO-1996001827-A1 TETRACYCLIC DERIVATIVES AND THEIR USE AS ANTITUMOUR AGENTS THE WELLCOME FOUNDATION LIMITED (GB) 1996-01-25 WO disclosed