SCHEMBL8537401

SCHEMBL8537401

O=Cc1nc(Br)c(Br)n1COCc1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.44
TSHR P16473 1/20 0.38
VDR P11473 2/20 0.33
MAPT P10636 2/20 0.33
RAB9A P51151 2/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
L3MBTL1 Q9Y468 2/20 0.33
NPC1 O15118 1/20 0.33
AR P10275 1/20 0.33
MAOA P21397 1/20 0.33
MAOB P27338 1/20 0.33
LMNA P02545 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
USP2 O75604 1/20 0.32
MAPK1 P28482 1/20 0.32
KDM4E B2RXH2 1/20 0.32
LTA4H P09960 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8536161 0.77 ALDH1A1 (0.43) ALDH1A1TSHRMAPTRAB9ASMN1; SMN2
SCHEMBL6928223 0.76 ALDH1A1 (0.45) ALDH1A1TSHRRAB9AL3MBTL1LMNA
SCHEMBL8532701 0.76 ALDH1A1 (0.42) ALDH1A1TSHRMAPTRAB9ASMN1; SMN2
SCHEMBL6922966 0.74 ALDH1A1 (0.43) ALDH1A1TSHRMAPTRAB9ASMN1; SMN2
SCHEMBL9593156 0.72 PDE4A (0.43) ALDH1A1
Hydrochloric Acid SCHEMBL8563542 0.71 ALDH1A1 (0.39) ALDH1A1TSHRMAPTRAB9ASMN1; SMN2
SCHEMBL20752451 0.69 BRD4 (0.44) ALDH1A1TSHRRAB9ASMN1; SMN2L3MBTL1
SCHEMBL6970946 0.69 TSHR (0.40) ALDH1A1TSHRMAPTRAB9ASMN1; SMN2
SCHEMBL6030662 0.68 KDM4E (0.52) ALDH1A1TSHRVDRMAPTRAB9A
SCHEMBL12650380 0.67 ALDH1A1 (0.50) ALDH1A1TSHRRAB9ASMN1; SMN2L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5719140-A ANALGESICS, PROSTAGLANDIN-E2 ANTAGONISTS G.D. SEARLE & CO. (US) 1998-02-17 US disclosed
EP-0696283-B1 2-, 3-, 4-, 5-, 6-, 7-, 8-, 9- AND/OR 10-SUBSTITUTED DIBENZOXAZEPINE COMPOUNDS, PHARMACEUTICAL COMPOSITIONS AND METHODS OF USE SEARLE & CO (US) 1997-09-17 EP disclosed
US-5395932-A Analgesics, prostaglandin E2 inhibitors G. D. SEARLE & CO. (US) 1995-03-07 US disclosed
WO-1994025456-A1 2-, 3-, 4-, 5-, 6-, 7-, 8-, 9- AND/OR 10-SUBSTITUTED DIBENZOXAZEPINE COMPOUNDS, PHARMACEUTICAL COMPOSITIONS AND METHODS OF USE G.D. SEARLE & CO. (US) 1994-11-10 WO disclosed