SCHEMBL8536161

SCHEMBL8536161

BrCc1nc(Br)c(Br)n1COCc1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.43
TSHR P16473 3/20 0.40
VCP P55072 1/20 0.34
TRPA1 O75762 1/20 0.33
L3MBTL1 Q9Y468 3/20 0.33
KDM4E B2RXH2 2/20 0.33
MAPK1 P28482 2/20 0.32
NPC1 O15118 1/20 0.32
LMNA P02545 1/20 0.32
TP53 P04637 1/20 0.32
POLB P06746 1/20 0.32
MAPT P10636 1/20 0.32
HTT P42858 1/20 0.32
RAB9A P51151 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
USP2 O75604 1/20 0.31
IDO1 P14902 1/20 0.31
CA1 P00915 2/20 0.30
CA2 P00918 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8532701 0.87 ALDH1A1 (0.42) ALDH1A1TSHRVCPL3MBTL1KDM4E
SCHEMBL6928223 0.87 ALDH1A1 (0.45) ALDH1A1TSHRVCPL3MBTL1MAPK1
SCHEMBL9593156 0.82 PDE4A (0.43) ALDH1A1POLB
SCHEMBL8537401 0.77 ALDH1A1 (0.44) ALDH1A1TSHRL3MBTL1KDM4EMAPK1
SCHEMBL6922966 0.70 ALDH1A1 (0.43) ALDH1A1TSHRVCPL3MBTL1MAPK1
SCHEMBL9051616 0.68 ALDH1A1 (0.40) ALDH1A1TSHRVCPL3MBTL1MAPK1
SCHEMBL4576525 0.66 ALDH1A1 (0.47) ALDH1A1TSHRL3MBTL1MAPK1NPC1
SCHEMBL12650380 0.66 ALDH1A1 (0.50) ALDH1A1TSHRL3MBTL1MAPK1NPC1
SCHEMBL1781279 0.66 ALDH1A1 (0.53) ALDH1A1TSHRL3MBTL1MAPK1NPC1
SCHEMBL12562962 0.65 ALDH1A1 (0.46) ALDH1A1TSHRVCPLMNARAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5719140-A ANALGESICS, PROSTAGLANDIN-E2 ANTAGONISTS G.D. SEARLE & CO. (US) 1998-02-17 US disclosed
EP-0696283-B1 2-, 3-, 4-, 5-, 6-, 7-, 8-, 9- AND/OR 10-SUBSTITUTED DIBENZOXAZEPINE COMPOUNDS, PHARMACEUTICAL COMPOSITIONS AND METHODS OF USE SEARLE & CO (US) 1997-09-17 EP disclosed
US-5395932-A Analgesics, prostaglandin E2 inhibitors G. D. SEARLE & CO. (US) 1995-03-07 US disclosed
WO-1994025456-A1 2-, 3-, 4-, 5-, 6-, 7-, 8-, 9- AND/OR 10-SUBSTITUTED DIBENZOXAZEPINE COMPOUNDS, PHARMACEUTICAL COMPOSITIONS AND METHODS OF USE G.D. SEARLE & CO. (US) 1994-11-10 WO disclosed