SCHEMBL6928223

SCHEMBL6928223

CCc1nc(Br)c(Br)n1COCc1ccccc1

nearest known ligand 0.45

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.45
RECQL P46063 1/20 0.40
TSHR P16473 2/20 0.39
VCP P55072 1/20 0.36
TLR7 Q9NYK1 1/20 0.35
LMNA P02545 2/20 0.34
L3MBTL1 Q9Y468 2/20 0.34
HTT P42858 1/20 0.34
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
RAB9A P51151 1/20 0.33
TP53 P04637 1/20 0.32
USP2 O75604 1/20 0.32
MAPK1 P28482 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8536161 0.87 ALDH1A1 (0.43) ALDH1A1TSHRVCPLMNAL3MBTL1
SCHEMBL9593156 0.87 PDE4A (0.43) ALDH1A1TLR7
SCHEMBL8532701 0.86 ALDH1A1 (0.42) ALDH1A1TSHRVCPLMNAL3MBTL1
SCHEMBL6922966 0.83 ALDH1A1 (0.43) ALDH1A1RECQLTSHRVCPTLR7
SCHEMBL8536407 0.82 ALDH1A1 (0.46) ALDH1A1RECQLTSHRVCPLMNA
SCHEMBL17005386 0.78 ALDH1A1 (0.43) ALDH1A1TSHRVCPLMNAHTT
SCHEMBL8537401 0.76 ALDH1A1 (0.44) ALDH1A1TSHRLMNAL3MBTL1RAB9A
Ethylene SCHEMBL6923915 0.74 ALDH1A1 (0.36) ALDH1A1RECQLVCP
SCHEMBL12650380 0.68 ALDH1A1 (0.50) ALDH1A1TSHRLMNAL3MBTL1MEN1
SCHEMBL8562859 0.67 ALDH1A1 (0.38) ALDH1A1RECQLTSHRVCPLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1140929-B1 1H-IMIDAZO 4,5-D]PYRIDAZIN-7-ONES, 3H-IMIDAZO 4,5-C]PYRIDIN-4-ONES AND CORRESPONDING THIONES AS CORTICOTROPIN RELEASING FACTOR (CRF) RECEPTOR LIGANDS BRISTOL MYERS SQUIBB PHARMA CO (US) 2003-10-15 EP disclosed
US-6518271-B1 1H-imidazo[4,5-d]pyridazin-7-one, and corresponding thiones as corticotropin releasing factor (CRF) receptor ligands BRISTOL-MYERS SQUIBB COMPANY 2003-02-11 US disclosed
US-6271380-B1 TREATING ANXIETY, DEPRESSION, AND OTHER PSYCHIATRIC, NEUROLOGICAL DISORDERS AS WELL IMMUNOLOGICAL, CARDIOVASCULAR OR HEART-RELATED DISEASES AND COLONIC HYPERSENSITIVITY ASSOCIATED WITH PSYCHOPATHOLOGICAL DISTURBANCE AND STRESS. DUPONT PHARMACEUTICALS COMPANY 2001-08-07 US disclosed