SCHEMBL8537553

SCHEMBL8537553

c1csc(Sc2ccccc2-c2ncc[nH]2)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CSNK1A1 P48729 1/20 0.41
TYRO3 Q06418 1/20 0.41
DYRK1B Q9Y463 1/20 0.41
NISCH Q9Y2I1 2/20 0.40
MTOR P42345 1/20 0.40
ADK P55263 1/20 0.40
GABRA1 P14867 1/20 0.38
GABRG2 P18507 1/20 0.38
GABRB3 P28472 1/20 0.38
GABRA5 P31644 1/20 0.38
GABRA3 P34903 1/20 0.38
GABRA2 P47869 1/20 0.38
IDO1 P14902 1/20 0.35
ADRA1A P35348 1/20 0.35
FBP1 P09467 1/20 0.34
SCN9A Q15858 1/20 0.34
MEN1 O00255 1/20 0.33
ALDH1A1 P00352 1/20 0.33
KMT2A Q03164 1/20 0.33
ADRA2A P08913 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11201564 0.73 FBP1 (0.42) NISCHMTORADKGABRA1GABRG2
SCHEMBL8537576 0.73 CSNK1A1 (0.49) CSNK1A1TYRO3DYRK1BNISCHMTOR
Hydrochloric Acid SCHEMBL20204146 0.72 CSNK1A1 (0.47) CSNK1A1TYRO3DYRK1BNISCHMTOR
SCHEMBL9287236 0.72 NISCH (0.64) CSNK1A1TYRO3DYRK1BNISCHMTOR
SCHEMBL14886257 0.70 NISCH (0.61) CSNK1A1TYRO3DYRK1BNISCHMTOR
SCHEMBL8536874 0.70 CSNK1A1 (0.45) CSNK1A1TYRO3DYRK1BNISCHMTOR
SCHEMBL8540626 0.70 CSNK1A1 (0.45) CSNK1A1TYRO3DYRK1BNISCHMTOR
SCHEMBL8538268 0.70 CSNK1A1 (0.45) CSNK1A1TYRO3DYRK1BNISCHMTOR
SCHEMBL10333561 0.69 KDM4E (0.55) IDO1MEN1ALDH1A1KMT2A
SCHEMBL8603493 0.68 F2RL1 (0.48) CSNK1A1TYRO3DYRK1BNISCHMTOR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0857171-A2 IMIDAZOLE DERIVATIVES AND THE USE THEREOF AS NITROGEN MONOXIDE SYNTHASE INHIBITORS SCHERING AKTIENGESELLSCHAFT (DE) 1998-08-12 EP disclosed
WO-1997015555-A2 IMIDAZOLE DERIVATIVES AND THE USE THEREOF AS NITROGEN MONOXIDE SYNTHASE INHIBITORS SCHERING AKTIENGESELLSCHAFT (DE) 1997-05-01 WO disclosed