SCHEMBL8538009

SCHEMBL8538009

CC(C(=O)O)c1csc(CBr)n1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SHMT1 P34896 3/20 0.35
SHMT2 P34897 3/20 0.35
CTSK P43235 1/20 0.33
GAA P10253 1/20 0.32
MEN1 O00255 1/20 0.32
POLB P06746 1/20 0.32
RAB9A P51151 1/20 0.32
KMT2A Q03164 1/20 0.32
MMP1 P03956 1/20 0.32
MMP2 P08253 1/20 0.32
MMP9 P14780 1/20 0.32
MMP13 P45452 1/20 0.32
PTGS1 P23219 4/20 0.32
PTGS2 P35354 4/20 0.32
AKR1C3 P42330 3/20 0.32
LMNA P02545 2/20 0.32
CYP2C9 P11712 2/20 0.32
CXCR1 P25024 2/20 0.32
CXCR2 P25025 2/20 0.32
AKR1C2 P52895 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5779345 0.80 KMT2A (0.38) GAAMEN1POLBRAB9AKMT2A
SCHEMBL29285032 0.78 HDAC3 (0.36) SHMT1SHMT2PTGS1PTGS2AKR1C3
SCHEMBL1758678 0.73 PI4KB (0.47) MEN1POLBRAB9AKMT2ALMNA
SCHEMBL24917646 0.73 SHMT1 (0.37) SHMT1SHMT2PTGS1PTGS2LMNA
SCHEMBL1565803 0.73 HSD17B10 (0.46) MEN1RAB9AKMT2ALMNAADRB3
Hydrochloric Acid SCHEMBL1758691 0.71 HSD17B10 (0.44) GAAMEN1RAB9AKMT2ALMNA
SCHEMBL743961 0.71 MMP13 (0.57) MMP1MMP2MMP9MMP13
SCHEMBL5516186 0.70 ALDH1A1 (0.40) GAAMEN1POLBRAB9AKMT2A
SCHEMBL18099911 0.70 PIK3CD (0.32) SHMT1SHMT2PTGS1PTGS2LMNA
SCHEMBL14721346 0.70 AKR1C3 (0.33) SHMT1SHMT2PTGS1PTGS2AKR1C3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5719140-A ANALGESICS, PROSTAGLANDIN-E2 ANTAGONISTS G.D. SEARLE & CO. (US) 1998-02-17 US disclosed
EP-0696283-B1 2-, 3-, 4-, 5-, 6-, 7-, 8-, 9- AND/OR 10-SUBSTITUTED DIBENZOXAZEPINE COMPOUNDS, PHARMACEUTICAL COMPOSITIONS AND METHODS OF USE SEARLE & CO (US) 1997-09-17 EP disclosed
US-5395932-A Analgesics, prostaglandin E2 inhibitors G. D. SEARLE & CO. (US) 1995-03-07 US disclosed
WO-1994025456-A1 2-, 3-, 4-, 5-, 6-, 7-, 8-, 9- AND/OR 10-SUBSTITUTED DIBENZOXAZEPINE COMPOUNDS, PHARMACEUTICAL COMPOSITIONS AND METHODS OF USE G.D. SEARLE & CO. (US) 1994-11-10 WO disclosed