SCHEMBL8538736

SCHEMBL8538736

CSCc1cccc(C(F)(F)F)c1F

nearest known ligand 0.40

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
AKR1B1 P15121 1/20 0.40
IDO1 P14902 2/20 0.38
P2RX7 Q99572 8/20 0.38
FFAR4 Q5NUL3 1/20 0.36
CD38 P28907 1/20 0.35
MPL P40238 2/20 0.35
CTSS P25774 1/20 0.35
EPHX2 P34913 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL515164 0.82 IDO1 (0.50) IDO1
SCHEMBL25870492 0.82 AKR1B1 (0.38) AKR1B1IDO1P2RX7FFAR4CD38
SCHEMBL6063364 0.80 IDO1 (0.41) IDO1P2RX7
SCHEMBL5415312 0.79 GABRA1 (0.46) AKR1B1IDO1P2RX7CD38CTSS
SCHEMBL41933 0.76 MAOB (0.47) AKR1B1IDO1P2RX7CD38MPL
SCHEMBL13551083 0.76 EPHX2 (0.40) AKR1B1IDO1P2RX7CD38CTSS
SCHEMBL17830317 0.76 AKR1B1 (0.40) AKR1B1IDO1P2RX7CD38MPL
SCHEMBL150130 0.75 IDO1 (0.46) AKR1B1IDO1P2RX7FFAR4MPL
SCHEMBL20560274 0.75 AKR1B1 (0.42) AKR1B1IDO1P2RX7FFAR4MPL
SCHEMBL1145792 0.75 MPO (0.36)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0857171-A2 IMIDAZOLE DERIVATIVES AND THE USE THEREOF AS NITROGEN MONOXIDE SYNTHASE INHIBITORS SCHERING AKTIENGESELLSCHAFT (DE) 1998-08-12 EP disclosed
WO-1997015555-A2 IMIDAZOLE DERIVATIVES AND THE USE THEREOF AS NITROGEN MONOXIDE SYNTHASE INHIBITORS SCHERING AKTIENGESELLSCHAFT (DE) 1997-05-01 WO disclosed