SCHEMBL25870492

SCHEMBL25870492

CC(C)(C)SCc1cccc(C(F)(F)F)c1F

nearest known ligand 0.39

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
AKR1B1 P15121 1/20 0.38
P2RX7 Q99572 8/20 0.36
IDO1 P14902 2/20 0.36
POLQ O75417 1/20 0.35
CD38 P28907 1/20 0.34
CTSS P25774 1/20 0.33
MPL P40238 1/20 0.33
FFAR4 Q5NUL3 1/20 0.33
EPHX2 P34913 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8538736 0.82 AKR1B1 (0.40) AKR1B1P2RX7IDO1CD38CTSS
SCHEMBL13791091 0.77 MEP1B (0.39)
SCHEMBL17830317 0.77 AKR1B1 (0.40) AKR1B1P2RX7IDO1CD38CTSS
SCHEMBL5415312 0.76 GABRA1 (0.46) AKR1B1P2RX7IDO1POLQCD38
SCHEMBL26017719 0.76 P2RX7 (0.42) AKR1B1P2RX7IDO1CD38CTSS
SCHEMBL13791152 0.75 HTR2A (0.43) IDO1
SCHEMBL18873928 0.74 AKR1B1 (0.39) AKR1B1P2RX7IDO1CD38CTSS
SCHEMBL41933 0.74 MAOB (0.47) AKR1B1P2RX7IDO1CD38MPL
SCHEMBL13551083 0.73 EPHX2 (0.40) AKR1B1P2RX7IDO1CD38CTSS
SCHEMBL15432484 0.72 P2RX7 (0.44) AKR1B1P2RX7IDO1CD38CTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023118250-A1 8-AZA QUINAZOLINES AS BRAIN-PENETRANT SOS1-INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2023-06-29 WO disclosed