SCHEMBL8538958

SCHEMBL8538958

CC(C)(C)NC(=O)N1Cc2ccccc2CC1[C@H](O)[C@@H](O)C1Cc2ccccc2CN1C(=O)NC(C)(C)C

nearest known ligand 0.49

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.49
CYP3A4 P08684 1/20 0.49
CYP2C19 P33261 1/20 0.49
OPRM1 P35372 10/20 0.45
OPRD1 P41143 10/20 0.45
OPRK1 P41145 6/20 0.41
TRPM8 Q7Z2W7 1/20 0.41
ACE P12821 2/20 0.39
DRD2 P14416 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8538954 1.00 POLB (0.49) POLBCYP3A4CYP2C19OPRM1OPRD1
SCHEMBL8538961 1.00 POLB (0.49) POLBCYP3A4CYP2C19OPRM1OPRD1
SCHEMBL7980018 0.80 POLB (0.59) POLBCYP3A4CYP2C19ACE
SCHEMBL8541519 0.80 PRMT5 (0.46) OPRD1ACE
SCHEMBL7966652 0.80 POLB (0.59) POLBCYP3A4CYP2C19ACE
SCHEMBL17572854 0.72 PRMT5 (0.42) OPRM1OPRD1OPRK1ACE
SCHEMBL9596147 0.71 POLB (0.65) POLBCYP3A4CYP2C19ACE
SCHEMBL18711805 0.71 POLB (0.65) POLBCYP3A4CYP2C19OPRM1OPRD1
SCHEMBL18711811 0.71 POLB (0.61) POLBCYP3A4CYP2C19OPRM1ACE
SCHEMBL21081936 0.70 RIPK1 (0.48) POLBCYP3A4CYP2C19OPRM1OPRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0839798-A2 Intermediates for preparating non-peptide retroviral protease inhibitors ABBOTT LABORATORIES (US) 1998-05-06 EP disclosed
US-5545750-A TREATING HUMAN IMMUNODEFICIENCY VIRUS ABBOTT LABORATORIES (US) 1996-08-13 US disclosed
US-5142056-A Human immunodeficiency virus protease inhibitor ABBOTT LABORATORIES (US) 1992-08-25 US disclosed