SCHEMBL8539558

SCHEMBL8539558

N#Cc1cccc(C(F)(F)F)c1-c1ncc[nH]1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 1/20 0.44
PDE4A P27815 1/20 0.38
PDE4B Q07343 1/20 0.38
PDE4C Q08493 1/20 0.38
PDE4D Q08499 1/20 0.38
AR P10275 5/20 0.37
MTOR P42345 2/20 0.37
ADK P55263 1/20 0.37
NISCH Q9Y2I1 1/20 0.37
PTGES O14684 1/20 0.35
SLC22A12 Q96S37 1/20 0.35
TRPA1 O75762 1/20 0.34
PIK3CD O00329 2/20 0.34
PIK3C2B O00750 2/20 0.34
PIK3CG P48736 1/20 0.34
PDK2 Q15119 1/20 0.34
MEN1 O00255 1/20 0.33
ALDH1A1 P00352 1/20 0.33
KMT2A Q03164 1/20 0.33
EGLN2 Q96KS0 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8540664 0.78 TAAR1 (0.48) TAAR1ARMTORADKNISCH
SCHEMBL5271255 0.74 ROCK2 (0.43) TAAR1PDE4APDE4BPDE4CPDE4D
SCHEMBL8536464 0.71 TAAR1 (0.45) TAAR1MTORADKNISCHPIK3CD
SCHEMBL9952337 0.70 TAAR1 (0.44) TAAR1MTORADKNISCHPTGES
SCHEMBL2651232 0.70 CSNK1A1 (0.49) PDE4APDE4BPDE4CPDE4DMTOR
SCHEMBL29360220 0.70 CSNK1A1 (0.49) TAAR1MTORADKNISCHTRPA1
SCHEMBL773131 0.70 CSNK1A1 (0.49) TAAR1MTORADKNISCHTRPA1
SCHEMBL7235096 0.70 TAAR1 (0.49) TAAR1MTORADKNISCHTRPA1
SCHEMBL20497275 0.69 LRRK2 (0.46) TAAR1PDE4APDE4BPDE4CPDE4D
SCHEMBL4765948 0.69 LRRK2 (0.44) PDE4APDE4BPDE4CPDE4DMTOR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0857171-A2 IMIDAZOLE DERIVATIVES AND THE USE THEREOF AS NITROGEN MONOXIDE SYNTHASE INHIBITORS SCHERING AKTIENGESELLSCHAFT (DE) 1998-08-12 EP disclosed
WO-1997015555-A2 IMIDAZOLE DERIVATIVES AND THE USE THEREOF AS NITROGEN MONOXIDE SYNTHASE INHIBITORS SCHERING AKTIENGESELLSCHAFT (DE) 1997-05-01 WO disclosed