SCHEMBL8539783

SCHEMBL8539783

Clc1nc(Nc2ccccc2)nc2nc[nH]c12

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK2 P24941 7/20 0.64
CDK1 P06493 3/20 0.64
NEK2 P51955 2/20 0.64
CHEK1 O14757 2/20 0.64
CDK7 P50613 2/20 0.64
AURKA O14965 1/20 0.64
CHEK2 O96017 1/20 0.64
ABL1 P00519 1/20 0.64
LCK P06239 1/20 0.64
FYN P06241 1/20 0.64
LYN P07948 1/20 0.64
MET P08581 1/20 0.64
SRC P12931 1/20 0.64
RPS6KB1 P23443 1/20 0.64
MAPK3 P27361 1/20 0.64
MAPK1 P28482 1/20 0.64
AKT2 P31751 1/20 0.64
CSNK1D P48730 1/20 0.64
GSK3B P49841 1/20 0.64
PLK1 P53350 1/20 0.64

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL459414 0.83 ADORA3 (0.68) CDK2CDK1NEK2CHEK1CDK7
SCHEMBL16147019 0.82 POLA1 (0.65) CDK2CDK1NEK2CHEK1CDK7
SCHEMBL16147002 0.82 CDK2 (0.64) CDK2CDK1NEK2CHEK1CDK7
SCHEMBL8369496 0.79 CDK1 (0.62) CDK2CDK1MAPK1POLA1ADORA3
SCHEMBL8539781 0.77 MAPK1 (0.50) CDK2CDK1NEK2CHEK1CDK7
SCHEMBL7112087 0.76 CDK2 (0.62) CDK2CDK1NEK2CHEK1CDK7
SCHEMBL3001381 0.76 TNNI3K (0.61) SRC
SCHEMBL27824249 0.76 DPP4 (0.61) CDK2POLA1ADORA3PDPK1
SCHEMBL5779077 0.74 POLA1 (0.60) CDK2NEK2POLA1PDPK1JAK2
SCHEMBL7666283 0.74 POLA1 (0.60) CDK2CDK1NEK2CDK7POLA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0794781-A4 DRUGS TO PREVENT RECURRENT HERPES VIRUS INFECTIONS UNIV MASSACHUSETTS MEDICAL (US) 1998-04-22 EP disclosed
EP-0794781-A1 DRUGS TO PREVENT RECURRENT HERPES VIRUS INFECTIONS UNIVERSITY OF MASSACHUSETTS MEDICAL CENTER (US) 1997-09-17 EP disclosed
US-5646155-A ADMINISTERING A 9-SUBSTITUTED-N2-PHENYLGUANINE DERIVATIVE UNIVERSITY OF MASSACHUSETTS MEDICAL CENTER (US) 1997-07-08 US disclosed
WO-1996020711-A1 DRUGS TO PREVENT RECURRENT HERPES VIRUS INFECTIONS UNIVERSITY OF MASSACHUSETTS MEDICAL CENTER (US) 1996-07-11 WO disclosed