SCHEMBL8539798

SCHEMBL8539798

CCc1cc(S(=O)(=O)C(CC)CC)c(C(F)(F)F)cc1C(=O)Cl

nearest known ligand 0.32

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 3/20 0.32
AKR1C2 P52895 3/20 0.32
DDR1 Q08345 1/20 0.30
GSTO1 P78417 1/20 0.30
CTSS P25774 1/20 0.30
CTSK P43235 1/20 0.30
AKR1B10 O60218 1/20 0.30
AKR1C4 P17516 1/20 0.30
AKR1C1 Q04828 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8539826 0.88 EGLN1 (0.30)
SCHEMBL8542335 0.88 EGLN1 (0.37) DDR1GSTO1
SCHEMBL8538459 0.87 AKR1C3 (0.33) AKR1C3AKR1C2DDR1GSTO1CTSS
SCHEMBL8538275 0.84 PSEN1 (0.30)
SCHEMBL8541620 0.83 DDR1 (0.39) DDR1
SCHEMBL8541505 0.82 DDR1 (0.32) DDR1GSTO1
SCHEMBL6935396 0.82 SLC9A1 (0.38)
SCHEMBL8542924 0.80 EGLN1 (0.40) DDR1
SCHEMBL8543032 0.80 SLC9A1 (0.33)
SCHEMBL8538912 0.78 CCR2 (0.34) DDR1CTSSCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1071743-C Sulfuryl or sulfinyl benzoyl guanidine derivative MERCK PATENT GMBH (DE) 2001-09-26 CN disclosed
US-5744641-A Sulfonyl- or sulfinylbenzoylguanidine derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1998-04-28 US disclosed
CN-1148590-A Sulfuryl or sulfinyl benzoyl guanidine derivative MERCK PATENT GMBH (DE) 1997-04-30 CN disclosed