SCHEMBL8540505

SCHEMBL8540505

O=C(CCc1ccccc1)N1CCC(CCO)CC1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.68
NPC1 O15118 1/20 0.63
TDP1 Q9NUW8 1/20 0.63
TSHR P16473 1/20 0.60
GRIN2B Q13224 1/20 0.60
CHRNB2 P17787 1/20 0.59
CHRNB4 P30926 1/20 0.59
CHRNA3 P32297 1/20 0.59
CHRNA4 P43681 1/20 0.59
FKBP1A P62942 1/20 0.58
FAAH O00519 1/20 0.58
HPGD P15428 1/20 0.54
SMN1; SMN2 Q16637 1/20 0.54
CHRM3 P20309 1/20 0.54
NAAA Q02083 1/20 0.54
L3MBTL1 Q9Y468 1/20 0.53
HDAC3 O15379 1/20 0.53
HDAC4 P56524 1/20 0.53
HDAC1 Q13547 1/20 0.53
HDAC7 Q8WUI4 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8542093 0.92 POLB (0.64) POLBNPC1TDP1TSHRGRIN2B
SCHEMBL8540623 0.88 POLB (0.71) POLBNPC1TDP1TSHRGRIN2B
SCHEMBL8541862 0.87 POLB (0.66) POLBNPC1TDP1TSHRGRIN2B
SCHEMBL8540143 0.86 MEN1 (0.52) POLBNPC1TDP1TSHRGRIN2B
SCHEMBL18106966 0.85 HDAC3 (0.66) POLBNPC1TSHRFAAHL3MBTL1
SCHEMBL18435561 0.85 POLB (0.71) POLBNPC1TDP1GRIN2BCHRNB2
SCHEMBL8539110 0.85 FAAH (0.64) POLBNPC1TDP1TSHRGRIN2B
SCHEMBL24043594 0.84 POLB (0.69) POLBNPC1TDP1TSHRGRIN2B
SCHEMBL5369484 0.84 POLB (0.69) POLBNPC1TDP1TSHRGRIN2B
SCHEMBL16591625 0.84 POLB (0.69) POLBNPC1TDP1TSHRGRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0705258-B1 AZOLYL-CYCLIC AMINE DERIVATIVES WITH IMMUNOMODULATORY ACTIVITY KNOLL AG (DE) 1998-12-30 EP disclosed
US-5741800-A ANTIINFLAMMATORY AGENT, ANTIALLERGENS KNOLL AKTIENGESELLACHAFT (DE) 1998-04-21 US disclosed
EP-0705258-A1 AZOLYL-CYCLIC AMINE DERIVATIVES WITH IMMUNOMODULATORY ACTIVITY Knoll AG (DE) 1996-04-10 EP disclosed
WO-1995000507-A1 AZOLYL-CYCLIC AMINE DERIVATIVES WITH IMMUNOMODULATORY ACTIVITY KNOLL AG (DE) 1995-01-05 WO disclosed