SCHEMBL8540522

SCHEMBL8540522

O=C(CCc1ccccc1)N1CCCC(CCl)C1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 1/20 0.68
SMN1; SMN2 Q16637 1/20 0.68
NPC1 O15118 1/20 0.62
TDP1 Q9NUW8 1/20 0.62
CHRNB2 P17787 4/20 0.60
CHRNA4 P43681 4/20 0.60
CHRNB4 P30926 3/20 0.60
CHRNA3 P32297 3/20 0.60
ALDH1A1 P00352 1/20 0.59
POLB P06746 1/20 0.56
NAAA Q02083 1/20 0.53
KDM4E B2RXH2 1/20 0.52
MAPK1 P28482 1/20 0.52
FKBP1A P62942 1/20 0.51
GRIN2B Q13224 1/20 0.48
CHRM3 P20309 1/20 0.48
MEN1 O00255 1/20 0.48
MAPT P10636 1/20 0.48
KMT2A Q03164 1/20 0.48
TACR3 P29371 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8546498 0.90 HPGD (0.65) HPGDSMN1; SMN2NPC1TDP1CHRNB2
SCHEMBL8540196 0.88 SMN1; SMN2 (0.70) HPGDSMN1; SMN2NPC1TDP1CHRNB2
SCHEMBL8545138 0.86 SMN1; SMN2 (0.67) HPGDSMN1; SMN2NPC1TDP1CHRNB2
SCHEMBL8540059 0.83 POLB (0.69) HPGDSMN1; SMN2NPC1TDP1CHRNB2
SCHEMBL17646360 0.81 ALDH1A1 (0.72) HPGDSMN1; SMN2NPC1TDP1CHRNB2
SCHEMBL12849241 0.81 HPGD (0.71) HPGDSMN1; SMN2NPC1TDP1CHRNB2
SCHEMBL7311015 0.81 ALDH1A1 (0.72) HPGDSMN1; SMN2NPC1TDP1CHRNB2
SCHEMBL8540140 0.78 HPGD (0.57) HPGDSMN1; SMN2NPC1TDP1CHRNB2
SCHEMBL25432319 0.78 NPC1 (0.93) HPGDSMN1; SMN2NPC1TDP1ALDH1A1
SCHEMBL3700679 0.78 NPC1 (1.00) HPGDSMN1; SMN2NPC1TDP1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0705258-B1 AZOLYL-CYCLIC AMINE DERIVATIVES WITH IMMUNOMODULATORY ACTIVITY KNOLL AG (DE) 1998-12-30 EP disclosed
US-5741800-A ANTIINFLAMMATORY AGENT, ANTIALLERGENS KNOLL AKTIENGESELLACHAFT (DE) 1998-04-21 US disclosed
EP-0705258-A1 AZOLYL-CYCLIC AMINE DERIVATIVES WITH IMMUNOMODULATORY ACTIVITY Knoll AG (DE) 1996-04-10 EP disclosed
WO-1995000507-A1 AZOLYL-CYCLIC AMINE DERIVATIVES WITH IMMUNOMODULATORY ACTIVITY KNOLL AG (DE) 1995-01-05 WO disclosed