SCHEMBL8540942

SCHEMBL8540942

CN(C)CCNc1ccc(NCCN(C)C)c2c1C(=O)c1ncc[n+]([O-])c1C2=O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TOP2B Q02880 2/20 0.38
CCR9 P51686 1/20 0.37
SLC40A1 Q9NP59 1/20 0.37
MALT1 Q9UDY8 1/20 0.36
CYP2C19 P33261 1/20 0.36
NQO1 P15559 1/20 0.36
ALDH1A1 P00352 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
KAT2B Q92831 2/20 0.36
TOP2A P11388 1/20 0.35
CDC25A P30304 1/20 0.34
CDC25B P30305 1/20 0.34
CDC25C P30307 1/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
HRH3 Q9Y5N1 1/20 0.34
NQO2 P16083 1/20 0.34
ATAD2 Q6PL18 1/20 0.33
EHMT2 Q96KQ7 1/20 0.33
IDO1 P14902 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8545624 0.85 ECE1 (0.37) MEN1KMT2A
SCHEMBL8546215 0.84 TOP2B (0.43) TOP2BSLC40A1MALT1NQO1ALDH1A1
SCHEMBL8543297 0.81 MEN1 (0.51) TOP2BNQO1ALDH1A1NPSR1TOP2A
SCHEMBL8545090 0.78 MALT1 (0.44) TOP2BMALT1NQO1ALDH1A1NPSR1
SCHEMBL9389581 0.76 IDO1 (0.49) TOP2BSLC40A1MALT1CYP2C19KAT2B
SCHEMBL4188736 0.75 MALT1 (0.49) TOP2BSLC40A1MALT1CYP2C19NQO1
Hydrochloric Acid SCHEMBL4197846 0.73 MALT1 (0.47) TOP2BSLC40A1MALT1CYP2C19NQO1
SCHEMBL7808635 0.71 KAT2B (0.41) NQO1KAT2BTOP2ANQO2
SCHEMBL8542449 0.71 TOP2B (0.49) TOP2BSLC40A1MALT1NQO1ALDH1A1
Hydrochloric Acid SCHEMBL8545200 0.70 TOP2B (0.48) TOP2BSLC40A1MALT1NQO1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0639183-B1 NITROGEN OXIDES OF AZA- AND DIAZA-ANTHRACENEDIONE DERIVATIVES, THEIR PREPARATION AND THEIR USE AS ANTITUMOR AGENTS BOEHRINGER MANNHEIM ITALIA (IT) 1998-07-01 EP disclosed
WO-1992015566-A1 NITROGEN OXIDES OF AZA- AND DIAZA-ANTHRACENEDIONE DERIVATIVES AS ANTITUMOR AGENTS BOEHRINGER MANNHEIM ITALIA S.P.A. (IT) 1992-09-17 WO disclosed