SCHEMBL8541963

SCHEMBL8541963

COC(=O)c1cc(C2OCCO2)cnc1C(=O)OC

nearest known ligand 0.37

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.37
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
KDM4E B2RXH2 4/20 0.36
ALDH1A1 P00352 3/20 0.36
OPRK1 P41145 10/20 0.35
NPSR1 Q6W5P4 1/20 0.34
HPGD P15428 1/20 0.34
HSD17B10 Q99714 1/20 0.34
GAA P10253 2/20 0.33
TSHR P16473 1/20 0.33
CFTR P13569 1/20 0.32
GLA P06280 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8546459 0.94 KDM4E (0.38) SMN1; SMN2NPC1RAB9AKDM4EALDH1A1
SCHEMBL8542643 0.94 KDM4E (0.38) SMN1; SMN2NPC1RAB9AKDM4EALDH1A1
SCHEMBL9724759 0.92 SMN1; SMN2 (0.35) SMN1; SMN2NPC1RAB9AKDM4EALDH1A1
SCHEMBL8542228 0.80
SCHEMBL8544532 0.76 KDM4E (0.40) SMN1; SMN2KDM4EALDH1A1NPSR1TSHR
SCHEMBL2487068 0.75 ATM (0.49) SMN1; SMN2KDM4EALDH1A1OPRK1NPSR1
SCHEMBL29833413 0.75 ATM (0.49) SMN1; SMN2KDM4EALDH1A1OPRK1NPSR1
SCHEMBL24411329 0.74 SYK (0.37) NPC1RAB9A
SCHEMBL24955122 0.74 MAPK1 (0.53) SMN1; SMN2NPC1RAB9AKDM4EALDH1A1
SCHEMBL27837816 0.73 OPRK1 (0.47) KDM4EALDH1A1OPRK1NPSR1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0434965-B1 Alkyl esters of 5-heterocyclic-pyridine-2,3-dicarboxylic acids and 5-heterocyclic 2-(2-imidazolin-2-yl) pyridines and methods for preparation thereof AMERICAN CYANAMID CO (US) 1998-05-20 EP claimed
EP-0434965-A2 Alkyl esters of 5-heterocyclic-pyridine-2,3-dicarboxylic acids and 5-heterocyclic 2-(2-imidazolin-2-yl) pyridines and methods for preparation thereof AMERICAN CYANAMID COMPANY (US) 1991-07-03 EP claimed
US-5026859-A Intermediates for herbicides AMERICAN CYANAMID COMPANY (US) 1991-06-25 US claimed
JP-4120074-A None JP disclosed
JP-H04120074-A 5-HETEROCYCLIC-PYRIDINE-2,3-DICARBOXYLIC ACID ALKYL ESTER, HIRBICIDAL 5-HETEROCYCLIC-2-(2-IMIDAZOLIN-2-YL)PYRIDINE AND THEIR PRODUCTION AMERICAN CYANAMID CO 1992-04-21 JP disclosed