SCHEMBL8546459

SCHEMBL8546459

COC(=O)c1cc(C2OCCCCO2)cnc1C(=O)OC

nearest known ligand 0.38

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.38
ALDH1A1 P00352 4/20 0.38
SMN1; SMN2 Q16637 3/20 0.38
HPGD P15428 2/20 0.38
HSD17B10 Q99714 2/20 0.38
OPRK1 P41145 11/20 0.36
CFTR P13569 1/20 0.36
NPC1 O15118 2/20 0.35
RAB9A P51151 2/20 0.35
ATM Q13315 1/20 0.34
POLB P06746 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8542643 0.97 KDM4E (0.38) KDM4EALDH1A1SMN1; SMN2HPGDHSD17B10
SCHEMBL8541963 0.94 SMN1; SMN2 (0.37) KDM4EALDH1A1SMN1; SMN2HPGDHSD17B10
SCHEMBL9724759 0.86 SMN1; SMN2 (0.35) KDM4EALDH1A1SMN1; SMN2HPGDHSD17B10
SCHEMBL8545598 0.77 KDM4E (0.38) KDM4EALDH1A1SMN1; SMN2HSD17B10
SCHEMBL8542228 0.75
SCHEMBL8544867 0.74 KDM4E (0.38) KDM4EALDH1A1SMN1; SMN2HSD17B10
SCHEMBL29833413 0.73 ATM (0.49) KDM4EALDH1A1SMN1; SMN2HSD17B10OPRK1
SCHEMBL2487068 0.73 ATM (0.49) KDM4EALDH1A1SMN1; SMN2HSD17B10OPRK1
SCHEMBL27837816 0.71 OPRK1 (0.47) KDM4EALDH1A1HPGDHSD17B10OPRK1
SCHEMBL18760423 0.71 NLRP3 (0.38) KDM4EALDH1A1HPGDHSD17B10NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0434965-B1 Alkyl esters of 5-heterocyclic-pyridine-2,3-dicarboxylic acids and 5-heterocyclic 2-(2-imidazolin-2-yl) pyridines and methods for preparation thereof AMERICAN CYANAMID CO (US) 1998-05-20 EP claimed
EP-0434965-A2 Alkyl esters of 5-heterocyclic-pyridine-2,3-dicarboxylic acids and 5-heterocyclic 2-(2-imidazolin-2-yl) pyridines and methods for preparation thereof AMERICAN CYANAMID COMPANY (US) 1991-07-03 EP claimed
US-5026859-A Intermediates for herbicides AMERICAN CYANAMID COMPANY (US) 1991-06-25 US claimed