SCHEMBL8543797

SCHEMBL8543797

CCCCNC(=O)Oc1ccc2c(c1)c(C)cn2NC(CC)c1ccncc1F

nearest known ligand 0.62

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
BCHE P06276 5/20 0.62
ACHE P22303 1/20 0.56
FAAH O00519 1/20 0.38
LIPE Q05469 1/20 0.38
ALDH1A1 P00352 1/20 0.36
KMT2A Q03164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8537927 0.97 BCHE (0.58) BCHEACHEFAAH
SCHEMBL8539761 0.89 ACHE (0.70) BCHEACHEALDH1A1
SCHEMBL8543197 0.87 BCHE (0.62) BCHEACHEFAAH
SCHEMBL9738851 0.86 BCHE (0.50) BCHEACHEFAAHLIPE
Hydrochloric Acid SCHEMBL9671998 0.85 BCHE (0.49) BCHEACHEFAAHLIPE
SCHEMBL9738706 0.83 BCHE (0.47) BCHEFAAH
Hydrochloric Acid SCHEMBL9671926 0.82 BCHE (0.46) BCHEFAAH
SCHEMBL8543795 0.82 BCHE (0.64) BCHEACHEFAAHLIPE
SCHEMBL9672315 0.80 BCHE (0.49) BCHEACHELIPE
SCHEMBL8537924 0.79 BCHE (0.60) BCHEACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5102891-A Useful for treating various memory dysfunctions such as alzheimer's disease HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1992-04-07 US claimed
EP-0468401-B1 1-(Substituted pyridinylamino)-1H-indol-5-yl substituted carbamates, a process for their preparation and their use as medicaments HOECHST MARION ROUSSEL INC (US) 1998-09-16 EP disclosed
US-5102891-A Useful for treating various memory dysfunctions such as alzheimer's disease HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1992-04-07 US disclosed
EP-0468401-A2 1-(Substituted pyridinylamino)-1H-indol-5-yl substituted carbamates, a process and intermediates for their preparation and their use as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1992-01-29 EP disclosed