SCHEMBL8544571

SCHEMBL8544571

O=C(CN1CCC[C@H]1C(=O)NC(=O)c1ccccc1)NCc1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.49
TP53 P04637 1/20 0.48
ALDH1A1 P00352 3/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
GAA P10253 1/20 0.47
F2 P00734 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47
FKBP1A P62942 2/20 0.47
ITGA4 P13612 1/20 0.46
ITGB7 P26010 1/20 0.46
MITF O75030 1/20 0.46
HDAC1 Q13547 2/20 0.46
HDAC2 Q92769 2/20 0.46
HDAC3 O15379 1/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2C9 P11712 1/20 0.46
PKM P14618 1/20 0.46
CYP2C19 P33261 1/20 0.46
PTGER4 P35408 1/20 0.45
USP2 O75604 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8543273 0.84 SMN1; SMN2 (0.55) ALDH1A1SMN1; SMN2GAANPSR1
SCHEMBL8544789 0.84 NPSR1 (0.47) ALDH1A1GAANPSR1
SCHEMBL8544794 0.84 NPSR1 (0.47) ALDH1A1GAANPSR1
SCHEMBL8543314 0.83 CTSK (0.53) ALDH1A1GAANPSR1
SCHEMBL8543316 0.83 CTSK (0.53) ALDH1A1GAANPSR1
SCHEMBL8543596 0.83 NPC1 (0.52) ALDH1A1SMN1; SMN2NPSR1CYP3A4CYP2C19
SCHEMBL8543591 0.83 NPC1 (0.52) ALDH1A1SMN1; SMN2NPSR1CYP3A4CYP2C19
SCHEMBL8543317 0.81 F2 (0.58) ALDH1A1SMN1; SMN2F2FKBP1ACYP3A4
SCHEMBL8544838 0.81 P2RX7 (0.56) ALDH1A1
SCHEMBL8549125 0.81 NPSR1 (0.48) ALDH1A1SMN1; SMN2NPSR1FKBP1AHDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0564924-B1 2-Oxoethyl derivatives as immunosuppressants BAYER AG (US) 1998-09-09 EP claimed
EP-0564924-A2 2-Oxoethyl derivatives as immunosuppressants Bayer Corporation (US) 1993-10-13 EP claimed
EP-0564924-B1 2-Oxoethyl derivatives as immunosuppressants BAYER AG (US) 1998-09-09 EP disclosed
US-5686424-A FOR TREATING INFLAMMATION MILES INC. (US) 1997-11-11 US disclosed
EP-0564924-A2 2-Oxoethyl derivatives as immunosuppressants Bayer Corporation (US) 1993-10-13 EP disclosed