SCHEMBL8544838

SCHEMBL8544838

O=C(CN1CCC[C@@H]1C(=O)NC(=O)c1ccccc1)NCC12CC3CC(CC(C3)C1)C2

nearest known ligand 0.56

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 8/20 0.56
ALDH1A1 P00352 2/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
HSD11B1 P28845 1/20 0.43
LMNA P02545 1/20 0.43
EPHX1 P07099 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8546685 0.86 HSD11B1 (0.54) ALDH1A1HSD11B1EPHX1
SCHEMBL8546679 0.86 HSD11B1 (0.54) ALDH1A1HSD11B1EPHX1
SCHEMBL8544843 0.85 P2RX7 (0.59) P2RX7ALDH1A1L3MBTL1
SCHEMBL8544264 0.83 HSD11B1 (0.46) P2RX7ALDH1A1HSD11B1LMNAEPHX1
SCHEMBL8544257 0.83 HSD11B1 (0.46) P2RX7ALDH1A1HSD11B1LMNAEPHX1
SCHEMBL8544571 0.81 HTT (0.49) ALDH1A1
SCHEMBL8549977 0.81 HSD11B1 (0.44) P2RX7ALDH1A1HSD11B1EPHX1
SCHEMBL8549532 0.80 KMT2A (0.53) HSD11B1
SCHEMBL8549527 0.80 KMT2A (0.53) HSD11B1
SCHEMBL8543273 0.79 SMN1; SMN2 (0.55) ALDH1A1LMNAEPHX1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0564924-B1 2-Oxoethyl derivatives as immunosuppressants BAYER AG (US) 1998-09-09 EP claimed
EP-0564924-A2 2-Oxoethyl derivatives as immunosuppressants Bayer Corporation (US) 1993-10-13 EP claimed
EP-0564924-B1 2-Oxoethyl derivatives as immunosuppressants BAYER AG (US) 1998-09-09 EP disclosed
US-5686424-A FOR TREATING INFLAMMATION MILES INC. (US) 1997-11-11 US disclosed
EP-0564924-A2 2-Oxoethyl derivatives as immunosuppressants Bayer Corporation (US) 1993-10-13 EP disclosed