SCHEMBL8545113

SCHEMBL8545113

CCc1c(C(=O)O)sc2cccc(N3CCN(CCc4ccc(Cl)cc4)CC3)c12

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 3/20 0.43
DRD4 P21917 1/20 0.43
SIGMAR1 Q99720 2/20 0.41
SMYD2 Q9NRG4 1/20 0.41
MEN1 O00255 1/20 0.41
ALDH1A1 P00352 1/20 0.41
KMT2A Q03164 1/20 0.41
EBP Q15125 1/20 0.40
ADRA1D P25100 5/20 0.39
ADRA1A P35348 5/20 0.39
ADRA1B P35368 5/20 0.39
HTR1A P08908 5/20 0.39
HTR2C P28335 1/20 0.39
CACNA1G O43497 1/20 0.39
HTR2A P28223 2/20 0.39
SLC6A4 P31645 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8546530 0.99 DRD2 (0.43) DRD2DRD4SIGMAR1SMYD2MEN1
SCHEMBL8545044 0.92 MEN1 (0.49) DRD2SIGMAR1MEN1ALDH1A1KMT2A
SCHEMBL8545232 0.91 MEN1 (0.44) DRD2MEN1ALDH1A1KMT2AADRA1D
Hydrochloric Acid SCHEMBL8545543 0.91 MEN1 (0.48) DRD2SIGMAR1MEN1ALDH1A1KMT2A
Hydrochloric Acid SCHEMBL8545099 0.90 MEN1 (0.43) DRD2MEN1ALDH1A1KMT2AADRA1D
SCHEMBL8549117 0.90 CYP2C9 (0.48) DRD2MEN1ALDH1A1KMT2AADRA1D
Hydrochloric Acid SCHEMBL8543414 0.90 CYP2C9 (0.47) DRD2MEN1ALDH1A1KMT2AADRA1D
SCHEMBL8551139 0.90 ADRA1D (0.52) SIGMAR1MEN1ALDH1A1KMT2AADRA1D
Hydrochloric Acid SCHEMBL8549071 0.89 ADRA1D (0.51) SIGMAR1MEN1ALDH1A1KMT2AADRA1D
SCHEMBL8544241 0.86 MEN1 (0.45) SIGMAR1MEN1ALDH1A1KMT2AHTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0660832-B1 SEROTONIN RECEPTOR AGENTS MERRELL PHARMA INC (US) 1998-01-14 EP disclosed
US-5436246-A Compounds for treatment of anxiety, depression, migraine, stroke, angina and hypertension MERRELL DOW PHARMACEUTICALS INC. 1995-07-25 US disclosed
EP-0660832-A1 SEROTONIN RECEPTOR AGENTS MERRELL PHARMACEUTICALS INC. (US) 1995-07-05 EP disclosed
WO-1994006789-A1 SEROTONIN RECEPTOR AGENTS MERRELL DOW PHARMACEUTICALS INC. (US) 1994-03-31 WO disclosed