SCHEMBL8551139

SCHEMBL8551139

CCc1c(C(=O)O)sc2cccc(N3CCN(CCc4ccc(OC)cc4)CC3)c12

nearest known ligand 0.52

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ADRA1D P25100 5/20 0.52
ADRA1A P35348 5/20 0.52
ADRA1B P35368 5/20 0.52
SIGMAR1 Q99720 2/20 0.47
HTR1A P08908 3/20 0.43
ALDH1A1 P00352 2/20 0.43
HRH3 Q9Y5N1 1/20 0.43
MEN1 O00255 1/20 0.43
POLB P06746 1/20 0.43
KMT2A Q03164 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
OPRM1 P35372 1/20 0.42
HTR2C P28335 1/20 0.42
HTR1D P28221 1/20 0.42
HTR1B P28222 1/20 0.42
KCNJ1 P48048 1/20 0.42
KCNH2 Q12809 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8549071 0.99 ADRA1D (0.51) ADRA1DADRA1AADRA1BSIGMAR1HTR1A
SCHEMBL8545044 0.91 MEN1 (0.49) ADRA1DADRA1AADRA1BSIGMAR1HTR1A
SCHEMBL8545232 0.90 MEN1 (0.44) ADRA1DADRA1AADRA1BHTR1AALDH1A1
Hydrochloric Acid SCHEMBL8545543 0.90 MEN1 (0.48) ADRA1DADRA1AADRA1BSIGMAR1HTR1A
Hydrochloric Acid SCHEMBL8545099 0.90 MEN1 (0.43) ADRA1DADRA1AADRA1BHTR1AALDH1A1
SCHEMBL8545113 0.90 DRD2 (0.43) ADRA1DADRA1AADRA1BSIGMAR1HTR1A
SCHEMBL8549117 0.90 CYP2C9 (0.48) ADRA1DADRA1AADRA1BHTR1AALDH1A1
Hydrochloric Acid SCHEMBL8543414 0.89 CYP2C9 (0.47) ADRA1DADRA1AADRA1BHTR1AALDH1A1
Hydrochloric Acid SCHEMBL8546530 0.89 DRD2 (0.43) ADRA1DADRA1AADRA1BSIGMAR1HTR1A
SCHEMBL8544241 0.85 MEN1 (0.45) SIGMAR1HTR1AALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0660832-B1 SEROTONIN RECEPTOR AGENTS MERRELL PHARMA INC (US) 1998-01-14 EP disclosed
US-5436246-A Compounds for treatment of anxiety, depression, migraine, stroke, angina and hypertension MERRELL DOW PHARMACEUTICALS INC. 1995-07-25 US disclosed
EP-0660832-A1 SEROTONIN RECEPTOR AGENTS MERRELL PHARMACEUTICALS INC. (US) 1995-07-05 EP disclosed
WO-1994006789-A1 SEROTONIN RECEPTOR AGENTS MERRELL DOW PHARMACEUTICALS INC. (US) 1994-03-31 WO disclosed