SCHEMBL8545347

SCHEMBL8545347

c1ccc(CCCN2CCC(CCn3cncn3)CC2)cc1

nearest known ligand 0.58

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 3/20 0.53
CCR3 P51677 1/20 0.53
HRH3 Q9Y5N1 4/20 0.52
GRIN2B Q13224 1/20 0.51
SLC6A4 P31645 1/20 0.48
SLC6A3 Q01959 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8539485 0.90 HRH3 (0.51) SIGMAR1CCR3HRH3GRIN2B
Hydrochloric Acid SCHEMBL8541843 0.89 HRH3 (0.50) SIGMAR1CCR3HRH3GRIN2B
SCHEMBL83059 0.80 SIGMAR1 (0.69) SIGMAR1CCR3HRH3GRIN2B
SCHEMBL6648239 0.80 CYP19A1 (0.62) SIGMAR1
SCHEMBL8540771 0.80 GRIN2B (0.58) SIGMAR1CCR3HRH3GRIN2BSLC6A4
SCHEMBL8546036 0.79 POLB (0.54) GRIN2B
SCHEMBL8542051 0.78 GRIN2B (0.54) SIGMAR1CCR3HRH3GRIN2BSLC6A4
SCHEMBL8538300 0.78 GRIN2B (0.54) SIGMAR1CCR3HRH3GRIN2B
SCHEMBL8545033 0.78 SIGMAR1 (0.53) SIGMAR1CCR3HRH3GRIN2BSLC6A4
Hydrochloric Acid SCHEMBL8546852 0.77 GRIN2B (0.53) SIGMAR1CCR3HRH3GRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0705258-B1 AZOLYL-CYCLIC AMINE DERIVATIVES WITH IMMUNOMODULATORY ACTIVITY KNOLL AG (DE) 1998-12-30 EP disclosed
US-5741800-A ANTIINFLAMMATORY AGENT, ANTIALLERGENS KNOLL AKTIENGESELLACHAFT (DE) 1998-04-21 US disclosed
EP-0705258-A1 AZOLYL-CYCLIC AMINE DERIVATIVES WITH IMMUNOMODULATORY ACTIVITY Knoll AG (DE) 1996-04-10 EP disclosed
WO-1995000507-A1 AZOLYL-CYCLIC AMINE DERIVATIVES WITH IMMUNOMODULATORY ACTIVITY KNOLL AG (DE) 1995-01-05 WO disclosed