SCHEMBL8545767

SCHEMBL8545767

Cc1ccc(S(=O)(=O)Oc2ccc(OS(=O)(=O)c3ccc(C)cc3)c3c2C(=O)c2ccncc2C3=O)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA P21397 1/20 0.41
MAOB P27338 1/20 0.41
CDC25B P30305 1/20 0.41
GAA P10253 4/20 0.40
KMT2A Q03164 3/20 0.40
MEN1 O00255 2/20 0.40
ESR1 P03372 1/20 0.40
ESR2 Q92731 1/20 0.40
ALDH1A1 P00352 3/20 0.40
MAPT P10636 5/20 0.39
TDP1 Q9NUW8 2/20 0.39
LMNA P02545 2/20 0.39
MAPK1 P28482 2/20 0.39
GFER P55789 1/20 0.38
KEAP1 Q14145 1/20 0.38
NFE2L2 Q16236 1/20 0.38
TP53 P04637 2/20 0.38
CYP3A4 P08684 2/20 0.38
CASP1 P29466 2/20 0.38
BLM P54132 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7817372 0.93 KMT2A (0.37) MAOAMAOBCDC25BGAAKMT2A
SCHEMBL7810136 0.93 CDC25B (0.41) MAOAMAOBCDC25BGAAKMT2A
SCHEMBL7804670 0.93 KMT2A (0.37) MAOAMAOBCDC25BGAAKMT2A
SCHEMBL7817293 0.93 CDC25B (0.41) MAOAMAOBCDC25BGAAKMT2A
SCHEMBL9194706 0.86 KMT2A (0.43) GAAKMT2AMEN1ESR1ESR2
SCHEMBL594052 0.83 VDR (0.54) GAAKMT2AMEN1ESR1ESR2
SCHEMBL7814683 0.81 PRKDC (0.39) GAAKMT2AMEN1ESR1ESR2
SCHEMBL7817471 0.79 KMT2A (0.39) GAAKMT2AMEN1ESR1ESR2
SCHEMBL5779910 0.78 KEAP1 (0.36) MAOBGAAALDH1A1MAPTTDP1
SCHEMBL7845722 0.78 ALDH1A1 (0.31) GAAKMT2AMEN1ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0639183-B1 NITROGEN OXIDES OF AZA- AND DIAZA-ANTHRACENEDIONE DERIVATIVES, THEIR PREPARATION AND THEIR USE AS ANTITUMOR AGENTS BOEHRINGER MANNHEIM ITALIA (IT) 1998-07-01 EP disclosed
WO-1992015566-A1 NITROGEN OXIDES OF AZA- AND DIAZA-ANTHRACENEDIONE DERIVATIVES AS ANTITUMOR AGENTS BOEHRINGER MANNHEIM ITALIA S.P.A. (IT) 1992-09-17 WO disclosed