SCHEMBL8545794

SCHEMBL8545794

Fc1ccc(C(CCCN2CCN(c3nc4cccc5c4n3CCC5)CC2)c2ccc(F)cc2)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCN5A Q14524 2/20 0.43
SLC6A9 P48067 1/20 0.42
DRD3 P35462 7/20 0.42
DRD2 P14416 6/20 0.42
HTR2A P28223 5/20 0.42
ADRA1A P35348 5/20 0.42
HRH1 P35367 5/20 0.42
OPRK1 P41145 5/20 0.42
SLC6A3 Q01959 5/20 0.42
OPRD1 P41143 4/20 0.42
ADORA3 P0DMS8 4/20 0.42
CYP3A4 P08684 3/20 0.42
CYP2D6 P10635 3/20 0.42
CYP1A2 P05177 3/20 0.42
MEN1 O00255 3/20 0.42
KMT2A Q03164 3/20 0.42
CYP2C9 P11712 2/20 0.42
MLNR O43193 2/20 0.42
USP2 O75604 2/20 0.42
LMNA P02545 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8545734 0.78 CYP2C9 (0.47) DRD2SLC6A3CYP2C9SIGMAR1HTR1A
SCHEMBL8543289 0.76 NPC1 (0.45) RAB9AMAPT
SCHEMBL8545991 0.76 LMNA (0.50) DRD3DRD2MEN1KMT2ALMNA
SCHEMBL8544059 0.74 MAPT (0.44) CYP1A2MEN1KMT2AUSP2LMNA
SCHEMBL8548519 0.73 MAPT (0.47) MEN1KMT2AUSP2TSHRMAPK1
Hydrochloric Acid SCHEMBL8550810 0.72 MAPT (0.46) MEN1KMT2AUSP2TSHRMAPK1
SCHEMBL8548303 0.71 RAB9A (0.45) HTR2ACYP1A2MEN1KMT2AUSP2
SCHEMBL8549930 0.71 MCL1 (0.46) CYP1A2MEN1KMT2ACYP2C9USP2
SCHEMBL8545797 0.70 SLC6A9 (0.42) SCN5ASLC6A9DRD3DRD2HTR2A
SCHEMBL8545733 0.70 CYP2D6 (0.47) OPRK1OPRD1CYP2D6LMNAOPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0700913-B1 5,6-dihydro-4H-imidazo(4,5,1-ij)quinolines, processes for their preparation, their use as medicaments, and intermediate compounds HOECHST MARION ROUSSEL INC (US) 1998-06-03 EP claimed
US-5500423-A ANALGESICS HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1996-03-19 US claimed
EP-0700913-B1 5,6-dihydro-4H-imidazo(4,5,1-ij)quinolines, processes for their preparation, their use as medicaments, and intermediate compounds HOECHST MARION ROUSSEL INC (US) 1998-06-03 EP disclosed
US-5563272-A ANALGESICS HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1996-10-08 US disclosed
US-5500423-A ANALGESICS HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1996-03-19 US disclosed
EP-0700913-A1 5,6-dihydro-4H-imidazo(4,5,1-ij)quinolines, processes for their preparation, their use as medicaments, and intermediate compounds HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1996-03-13 EP disclosed