SCHEMBL8545893

SCHEMBL8545893

CC(C)(C)C(=O)CN1C(=O)CN=C(n2nccn2)c2ccccc21

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.46
KDM4E B2RXH2 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
MAPT P10636 2/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2C19 P33261 1/20 0.40
RECQL P46063 1/20 0.40
GAA P10253 1/20 0.40
HTT P42858 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
GPR55 Q9Y2T6 1/20 0.40
POLB P06746 1/20 0.39
HCRTR2 O43614 1/20 0.39
HDAC3 O15379 1/20 0.39
HDAC1 Q13547 1/20 0.39
HDAC8 Q9BY41 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
TP53 P04637 2/20 0.38
THRB P10828 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6940855 0.79 SMN1; SMN2 (0.64) ALDH1A1KDM4ESMN1; SMN2MAPTCYP1A2
SCHEMBL4992176 0.78 CYP1A2 (0.59) ALDH1A1KDM4ESMN1; SMN2MAPTCYP1A2
SCHEMBL6934431 0.76 SMN1; SMN2 (0.55) ALDH1A1KDM4ESMN1; SMN2MAPTCYP1A2
SCHEMBL8549514 0.76 CYP1A2 (0.46) ALDH1A1KDM4ESMN1; SMN2MAPTCYP1A2
SCHEMBL8548821 0.76 CYP1A2 (0.48) ALDH1A1KDM4ESMN1; SMN2MAPTCYP1A2
SCHEMBL8547276 0.76 ALDH1A1 (0.42) ALDH1A1KDM4ESMN1; SMN2MAPTCYP1A2
SCHEMBL8543118 0.75 KDM4E (0.45) ALDH1A1KDM4ESMN1; SMN2MAPTCYP1A2
SCHEMBL8546479 0.74 KDM4E (0.46) ALDH1A1KDM4ESMN1; SMN2MAPTCYP1A2
SCHEMBL7069966 0.71 TP53 (0.64) ALDH1A1SMN1; SMN2MAPTCYP1A2NPSR1
Urethane SCHEMBL8606798 0.70 CYP1A2 (0.51) ALDH1A1KDM4ESMN1; SMN2MAPTCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0715624-B1 PROCESS FOR THE PREPARATION OF BENZODIAZEPINE COMPOUNDS USEFUL AS ANTAGONISTS OF CCK OR OF GASTRINE YAMANOUCHI PHARMA CO LTD (JP) 1998-04-08 EP disclosed