SCHEMBL8546243

SCHEMBL8546243

N#CC(Cl)Cl.c1cc2ccc1-2

nearest known ligand 0.60

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.60
CYP3A4 P08684 2/20 0.60
ALOX15 P16050 1/20 0.60
HIF1A Q16665 1/20 0.60
MMP3 P08254 1/20 0.36
KIF11 P52732 2/20 0.32
PDPK1 O15530 1/20 0.31
ESR1 P03372 2/20 0.31
ESR2 Q92731 2/20 0.31
TRPA1 O75762 1/20 0.31
TSHR P16473 1/20 0.31
CYP1A2 P05177 1/20 0.30
TP53 P04637 1/20 0.30
TDP1 Q9NUW8 1/20 0.30
CA12 O43570 1/20 0.30
CA1 P00915 1/20 0.30
CA2 P00918 1/20 0.30
CA9 Q16790 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1180554 0.78
SCHEMBL2005231 0.73 ALDH1A1 (0.90) ALDH1A1CYP3A4ALOX15HIF1ATSHR
SCHEMBL28133271 0.73
SCHEMBL27898352 0.73 ALDH1A1 (0.60) ALDH1A1CYP3A4MMP3KIF11ESR1
SCHEMBL11080419 0.73 KIF11 (0.37) ALDH1A1CYP3A4MMP3KIF11ESR1
SCHEMBL11029698 0.73 ALDH1A1 (0.50) ALDH1A1CYP3A4ALOX15HIF1A
SCHEMBL11675959 0.69 ESR1 (0.39) ALDH1A1CYP3A4MMP3KIF11ESR1
Water SCHEMBL8153073 0.68
Acetonitrile SCHEMBL8836994 0.67 ALDH1A1 (0.75) ALDH1A1CYP3A4ALOX15HIF1ATSHR
Methyl Alcohol SCHEMBL28639463 0.67

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0474561-B1 Arylalkylamines, process for their preparation and pharmaceutical compositions containing them SANOFI SA (FR) 1998-12-09 EP disclosed
EP-0220112-B1 AROMATIC DERIVATIVES SUBSTITUTED BY AN (OMEGA-AMINO)-ALKANOL GROUP WITH AN ANTIMICROBIAL ACTIVITY, THEIR PREPARATION AND COMPOSITIONS CONTAINING THEM ELF SANOFI (FR) 1992-04-08 EP disclosed
EP-0474561-A1 Arylalkylamines, process for their preparation and pharmaceutical compositions containing them SANOFI (FR) 1992-03-11 EP disclosed
EP-0288352-B1 AROMATIC DERIVATIVES, THEIR PREPARATION AND THEIR USE AS ANTIMICROBICS SANOFI (FR) 1991-09-18 EP disclosed
EP-0288352-A1 Aromatic derivatives, their preparation and their use as antimicrobics SANOFI (FR) 1988-10-26 EP disclosed