SCHEMBL8546874

SCHEMBL8546874

O=C(c1ccc(CBr)cc1)c1cccc(C(=O)c2ccc(CBr)cc2)c1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 1/20 0.60
CES1 P23141 1/20 0.60
ATM Q13315 1/20 0.59
TDP1 Q9NUW8 1/20 0.59
L3MBTL1 Q9Y468 1/20 0.59
PBRM1 Q86U86 1/20 0.46
ALDH1A1 P00352 1/20 0.44
SRD5A2 P31213 3/20 0.44
MEN1 O00255 1/20 0.42
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
KMT2A Q03164 1/20 0.42
CLK1 P49759 1/20 0.42
DYRK1A Q13627 1/20 0.42
DYRK1B Q9Y463 1/20 0.42
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
CA9 Q16790 1/20 0.41
HSD17B1 P14061 1/20 0.41
HSD17B2 P37059 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20836220 0.92 CES2 (0.56) CES2CES1ATMTDP1L3MBTL1
SCHEMBL2931832 0.88 CES2 (0.51) CES2CES1ATMTDP1L3MBTL1
SCHEMBL118227 0.88 CES2 (0.77) CES2CES1ATMTDP1L3MBTL1
SCHEMBL9541276 0.87 CES2 (0.61) CES2CES1ALDH1A1SRD5A2KMT2A
SCHEMBL187134 0.87 CES2 (0.61) CES2CES1ALDH1A1SRD5A2KMT2A
SCHEMBL507406 0.84 GSK3B (0.60) CES2CES1
SCHEMBL185962 0.83 ATM (0.52) CES2CES1ATMTDP1L3MBTL1
SCHEMBL29572523 0.83 ATM (0.52) CES2CES1ATMTDP1L3MBTL1
SCHEMBL435297 0.82 L3MBTL1 (0.63) CES2CES1ATMTDP1L3MBTL1
SCHEMBL9151945 0.82 CES2 (0.69) CES2CES1ATMTDP1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0696585-B1 NOVEL BISOXADIAZOLIDINE DERIVATIVE YAMANOUCHI PHARMA CO LTD (JP) 1998-12-16 EP disclosed
US-5643931-A ANTIDIABETIC AGENTS YAMANOUCHI PHARMACEUTICAL CO., LTD. (JP) 1997-07-01 US disclosed
EP-0696585-A1 NOVEL BISOXADIAZOLIDINE DERIVATIVE YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 1996-02-14 EP disclosed