SCHEMBL8547847

SCHEMBL8547847

c1ccc2nc3ccc4c[nH]nc4c3cc2c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.46
ALDH1A1 P00352 2/20 0.46
GLA P06280 2/20 0.46
HPGD P15428 2/20 0.46
GAA P10253 2/20 0.46
RAB9A P51151 2/20 0.46
POLB P06746 2/20 0.46
KDM4E B2RXH2 2/20 0.46
NPC1 O15118 1/20 0.46
LMNA P02545 1/20 0.46
PTBP1 P26599 1/20 0.46
RCE1 Q9Y256 1/20 0.46
MAPT P10636 2/20 0.45
ACHE P22303 1/20 0.45
HTR3A P46098 1/20 0.40
ESR1 P03372 2/20 0.37
ESR2 Q92731 2/20 0.37
KDM1A O60341 1/20 0.36
PDE2A O00408 1/20 0.36
PDE3B Q13370 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1325210 0.77 ALDH1A1 (0.60) KMT2AALDH1A1GLAHPGDGAA
SCHEMBL5201632 0.76 ALDH1A1 (0.46) KMT2AALDH1A1HPGDRAB9APOLB
SCHEMBL4299906 0.75 ALDH1A1 (0.70) KMT2AALDH1A1GLAHPGDGAA
SCHEMBL15271630 0.75 ALDH1A1 (0.41) ALDH1A1HPGDGAAKDM4EACHE
SCHEMBL31465209 0.74 MAPT (0.56) KMT2AALDH1A1GLAHPGDGAA
SCHEMBL28424829 0.74 MAPT (0.56) KMT2AALDH1A1GLAHPGDGAA
SCHEMBL6032927 0.72 LMNA (0.59) KMT2AALDH1A1GLAHPGDGAA
SCHEMBL29712310 0.72 ALDH1A1 (0.58) KMT2AALDH1A1GLAHPGDGAA
SCHEMBL11690096 0.72 ALDH1A1 (0.58) KMT2AALDH1A1GLAHPGDGAA
SCHEMBL30853545 0.72 ALDH1A1 (0.58) KMT2AALDH1A1GLAHPGDGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0560231-B1 Pyrazolo(3,4-a)acridine derivatives as analgesics HOECHST MARION ROUSSEL INC (US) 1998-06-03 EP disclosed
EP-0560231-A1 Pyrazolo(3,4-a)acridine derivatives as analgesics HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1993-09-15 EP disclosed