SCHEMBL5201632

SCHEMBL5201632

c1ccc2c(c1)ccc1c[nH]nc12

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.46
CYP2A6 P11509 3/20 0.46
HSD17B10 Q99714 2/20 0.46
TDP1 Q9NUW8 2/20 0.46
TSHR P16473 2/20 0.46
NPC1 O15118 4/20 0.44
RAB9A P51151 4/20 0.44
HPRT1 P00492 1/20 0.42
HIF1A Q16665 1/20 0.39
CYP1B1 Q16678 1/20 0.39
MAPT P10636 4/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
KDM4E B2RXH2 2/20 0.38
HPGD P15428 2/20 0.38
TP53 P04637 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
MEN1 O00255 2/20 0.37
POLB P06746 2/20 0.37
KMT2A Q03164 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15271630 0.77 ALDH1A1 (0.41) ALDH1A1CYP2A6HSD17B10TDP1HPRT1
SCHEMBL8547847 0.76 KMT2A (0.46) ALDH1A1NPC1RAB9AMAPTKDM4E
SCHEMBL10667809 0.75 LMNA (0.59) ALDH1A1TDP1TSHRNPC1RAB9A
SCHEMBL8763443 0.74 ALDH1A1 (0.52) ALDH1A1CYP2A6HSD17B10TDP1TSHR
SCHEMBL4955116 0.74 IMPDH2 (0.42) KDM4ECYP3A4HTTCYP1A2
Iodide SCHEMBL10698948 0.74 LMNA (0.58) ALDH1A1TDP1TSHRNPC1RAB9A
SCHEMBL6070437 0.72 KIF11 (0.56) ALDH1A1HSD17B10TSHRMAPTKDM4E
SCHEMBL1727666 0.72 KDM4E (0.52) KDM4ECYP1A2
SCHEMBL5657095 0.72 LMNA (0.51) ALDH1A1HSD17B10TDP1TSHRHIF1A
SCHEMBL5741090 0.72 KDM4E (0.52) ALDH1A1HSD17B10TDP1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0724572-A1 FUSED TRICYCLIC HETEROAROMATIC DERIVATIVES AS DOPAMINE RECEPTOR SUBTYPE LIGANDS MERCK SHARP & DOHME LTD. (GB) 1996-08-07 EP claimed
WO-2021016670-A1 ANTIVIRAL AGENTS AND USES THEREOF GRIFFITH UNIVERSITY (AU) 2021-02-04 WO disclosed
EP-1339700-B1 PROCESS FOR THE PREPARATION OF BENZOTRIAZOLES CIBA SC HOLDING AG (CH) 2007-11-21 EP disclosed
EP-0724572-A1 FUSED TRICYCLIC HETEROAROMATIC DERIVATIVES AS DOPAMINE RECEPTOR SUBTYPE LIGANDS MERCK SHARP & DOHME LTD. (GB) 1996-08-07 EP disclosed