SCHEMBL8548510

SCHEMBL8548510

N=C(N)Nc1cccnn1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GOT1 P17174 1/20 0.55
FFAR2 O15552 1/20 0.40
P2RX7 Q99572 1/20 0.39
SIRT2 Q8IXJ6 1/20 0.38
CHRM2 P08172 1/20 0.35
CHRM4 P08173 1/20 0.35
CHRM1 P11229 1/20 0.35
CHRM3 P20309 1/20 0.35
FAAH O00519 6/20 0.34
JAK2 O60674 2/20 0.34
JAK1 P23458 2/20 0.34
TYK2 P29597 2/20 0.34
FPR2 P25090 1/20 0.34
LRRK2 Q5S007 1/20 0.34
JAK3 P52333 1/20 0.33
LCK P06239 1/20 0.33
CSNK1D P48730 1/20 0.32
CSNK1E P49674 1/20 0.32
AHR P35869 1/20 0.32
CYP1A2 P05177 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10622224 0.80 GOT1 (0.55) GOT1FFAR2P2RX7SIRT2CHRM2
SCHEMBL3988243 0.76
SCHEMBL2226467 0.73 RAB9A (0.59) CYP1A2
SCHEMBL15348825 0.73 GOT1 (0.52) GOT1FFAR2P2RX7SIRT2CHRM2
SCHEMBL14120037 0.73 GOT1 (0.57) GOT1FFAR2P2RX7SIRT2CHRM2
SCHEMBL10846209 0.72 GOT1 (0.50) GOT1FFAR2P2RX7SIRT2CHRM2
SCHEMBL1430882 0.72 GOT1 (0.50) GOT1FFAR2P2RX7SIRT2CHRM2
SCHEMBL697154 0.72
SCHEMBL29044120 0.72
SCHEMBL26520592 0.71 GOT1 (0.41) GOT1FFAR2P2RX7SIRT2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0825187-A1 Condensed pyridazinyl guanidines, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-02-25 EP disclosed
EP-0825187-A1 Condensed pyridazinyl guanidines, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-02-25 EP disclosed