SCHEMBL8548566

SCHEMBL8548566

COc1ccc(C2CCN(CCN(C)C(=O)c3ccc4c(c3)CCOC4)CC2)cc1

nearest known ligand 0.44

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 1/20 0.44
DRD2 P14416 5/20 0.44
MCHR1 Q99705 7/20 0.42
DRD4 P21917 3/20 0.41
HTR1D P28221 4/20 0.41
HTR2A P28223 4/20 0.41
HTR1A P08908 3/20 0.41
TNKS O95271 2/20 0.41
TNKS2 Q9H2K2 2/20 0.41
FASN P49327 1/20 0.40
PARP1 P09874 1/20 0.40
PARP2 Q9UGN5 1/20 0.40
SIGMAR1 Q99720 1/20 0.40
HTR1B P28222 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8549845 0.89 HRH3 (0.49) OPRM1DRD2MCHR1SIGMAR1
SCHEMBL8549609 0.86 DRD4 (0.58) DRD2DRD4HTR1DHTR2AHTR1A
SCHEMBL8549415 0.77 DRD4 (0.49) DRD2DRD4HTR1DHTR2AHTR1A
SCHEMBL8549485 0.76 DRD4 (0.48) DRD2DRD4HTR1DHTR2AHTR1A
SCHEMBL8550263 0.76 DRD4 (0.48) DRD2DRD4HTR1DHTR2AHTR1A
SCHEMBL8550144 0.75 DRD2 (0.50) DRD2DRD4HTR1DHTR2AHTR1A
SCHEMBL8550687 0.75 DRD4 (0.48) DRD2DRD4HTR1DHTR2AHTR1A
SCHEMBL8551575 0.75 DRD4 (0.48) DRD2DRD4HTR1DHTR2AHTR1A
SCHEMBL8549471 0.75 DRD4 (0.48) DRD2DRD4HTR1DHTR2AHTR1A
SCHEMBL8553551 0.75 DRD4 (0.48) DRD2DRD4HTR1DHTR2AHTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0836599-A1 1,6-DISUBSTITUTED ISOCHROMANS FOR TREATMENT OF MIGRAINE HEADACHES PHARMACIA & UPJOHN COMPANY (US) 1998-04-22 EP claimed
EP-0836599-A1 1,6-DISUBSTITUTED ISOCHROMANS FOR TREATMENT OF MIGRAINE HEADACHES PHARMACIA & UPJOHN COMPANY (US) 1998-04-22 EP disclosed