SCHEMBL8549845

SCHEMBL8549845

CN(CCN1CCC(c2ccccc2)CC1)C(=O)c1ccc2c(c1)CCOC2

nearest known ligand 0.49

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 2/20 0.49
MCHR1 Q99705 8/20 0.48
SIGMAR1 Q99720 1/20 0.43
SLC18A3 Q16572 2/20 0.42
DRD2 P14416 2/20 0.41
OPRM1 P35372 1/20 0.41
HTT P42858 1/20 0.40
KDM1A O60341 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8548566 0.89 OPRM1 (0.44) MCHR1SIGMAR1DRD2OPRM1
SCHEMBL8550173 0.81 MCHR1 (0.50) MCHR1SIGMAR1DRD2OPRM1KDM1A
SCHEMBL8551575 0.78 DRD4 (0.48) HRH3DRD2
SCHEMBL8553551 0.78 DRD4 (0.48) HRH3DRD2
SCHEMBL8549471 0.78 DRD4 (0.48) HRH3DRD2
SCHEMBL8550687 0.78 DRD4 (0.48) HRH3DRD2
SCHEMBL8550252 0.77 DRD4 (0.59) HRH3DRD2
SCHEMBL8550057 0.77 DRD4 (0.48) MCHR1HTT
SCHEMBL8550036 0.77 DRD4 (0.47) HRH3DRD2HTT
SCHEMBL8549100 0.77 DRD4 (0.47) HRH3DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0836599-A1 1,6-DISUBSTITUTED ISOCHROMANS FOR TREATMENT OF MIGRAINE HEADACHES PHARMACIA & UPJOHN COMPANY (US) 1998-04-22 EP claimed
EP-0836599-A1 1,6-DISUBSTITUTED ISOCHROMANS FOR TREATMENT OF MIGRAINE HEADACHES PHARMACIA & UPJOHN COMPANY (US) 1998-04-22 EP disclosed