SCHEMBL8548654

SCHEMBL8548654

CCOC(=O)c1cc2c(N3CCNCC3)cccc2s1

nearest known ligand 0.45

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MAPT P10636 1/20 0.43
LMNA P02545 1/20 0.42
KDM4E B2RXH2 1/20 0.42
TSHR P16473 1/20 0.42
HSD17B10 Q99714 1/20 0.42
HTR1A P08908 2/20 0.41
DRD2 P14416 1/20 0.41
DRD4 P21917 1/20 0.41
HTR2A P28223 1/20 0.41
HTR2C P28335 1/20 0.41
DRD3 P35462 1/20 0.41
SLC6A4 P31645 1/20 0.41
HTR5A P47898 1/20 0.41
F9 P00740 1/20 0.40
HTR6 P50406 1/20 0.40
ADRB1 P08588 1/20 0.40
THRB P10828 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8548772 0.99 MAPT (0.43) MAPTLMNAKDM4ETSHRHSD17B10
SCHEMBL8549470 0.87 MAPT (0.46) MAPTLMNAKDM4ETSHRHSD17B10
SCHEMBL17996841 0.85 ALDH1A1 (0.47) MAPTLMNAKDM4ETSHRHSD17B10
SCHEMBL17996836 0.84 MAPT (0.46) MAPTLMNAKDM4ETSHRHSD17B10
SCHEMBL8544023 0.84 HTR1A (0.48) MAPTLMNATSHRHSD17B10HTR1A
Hydrochloric Acid SCHEMBL6017128 0.84 HTR1A (0.47) MAPTLMNATSHRHSD17B10HTR1A
SCHEMBL9206773 0.83 KDM4E (0.38) MAPTLMNAKDM4ETSHRHSD17B10
SCHEMBL17080814 0.83 MAPT (0.49) MAPTLMNA
SCHEMBL8545029 0.82 CYP2D6 (0.38) MAPTLMNAKDM4ETSHRHSD17B10
SCHEMBL8545092 0.82 PRMT1 (0.57) MAPTLMNAHTR1ADRD2DRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0660832-B1 SEROTONIN RECEPTOR AGENTS MERRELL PHARMA INC (US) 1998-01-14 EP disclosed
US-5436246-A Compounds for treatment of anxiety, depression, migraine, stroke, angina and hypertension MERRELL DOW PHARMACEUTICALS INC. 1995-07-25 US disclosed
EP-0660832-A1 SEROTONIN RECEPTOR AGENTS MERRELL PHARMACEUTICALS INC. (US) 1995-07-05 EP disclosed
WO-1994006789-A1 SEROTONIN RECEPTOR AGENTS MERRELL DOW PHARMACEUTICALS INC. (US) 1994-03-31 WO disclosed