SCHEMBL8548718

SCHEMBL8548718

O=CNC(C(NC(=O)OCc1ccccc1)C(=O)O)[C@H]1CC(CCCCN[C@@H]2N=CCN2)=NO1

nearest known ligand 0.41

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 17/20 0.41
ITGAV P06756 13/20 0.41
ITGA2B P08514 13/20 0.41
CASP1 P29466 1/20 0.35
CASP3 P42574 1/20 0.35
CASP7 P55210 1/20 0.35
CASP6 P55212 1/20 0.35
CASP8 Q14790 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8551009 0.79 ITGB3 (0.45) ITGB3ITGAVITGA2B
SCHEMBL7402861 0.78 ITGB3 (0.67) ITGB3ITGAVITGA2B
SCHEMBL8644840 0.72 ATM (0.33) ITGB3ITGAVITGA2BCASP1CASP3
SCHEMBL7373306 0.72 GLS (0.39) ITGB3ITGAVITGA2B
SCHEMBL7400652 0.70 ITGB3 (0.67) ITGB3ITGAVITGA2B
SCHEMBL8643943 0.69 ITGB3 (0.36) ITGB3ITGAVITGA2B
SCHEMBL8177321 0.67 ITGB3 (0.42) ITGB3ITGAVITGA2B
SCHEMBL8546573 0.65 ITGB3 (0.49) ITGB3ITGAVITGA2B
SCHEMBL7406112 0.64 ITGB3 (0.65) ITGB3ITGAVITGA2B
SCHEMBL7396575 0.64 ITGB3 (0.43) ITGB3ITGAVITGA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0828737-A1 ISOXAZOLINE AND ISOXAZOLE DERIVATIVES AS INTEGRIN RECEPTOR ANTAGONISTS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1998-03-18 EP disclosed