SCHEMBL8548778

SCHEMBL8548778

O=[N+]([O-])c1cccc2c(-c3ccccc3)nnc(Cl)c12

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.47
MEN1 O00255 3/20 0.47
TDP1 Q9NUW8 4/20 0.43
ALDH1A1 P00352 6/20 0.42
MAPT P10636 3/20 0.42
LMNA P02545 1/20 0.42
GAA P10253 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
KDM4E B2RXH2 2/20 0.41
ABCG2 Q9UNQ0 1/20 0.40
OPRK1 P41145 1/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
MAPK1 P28482 2/20 0.40
RAB9A P51151 1/20 0.40
FBP1 P09467 1/20 0.39
ABCB1 P08183 1/20 0.38
ABCC1 P33527 1/20 0.38
POLB P06746 1/20 0.38
PDE5A O76074 1/20 0.37
CYP1A2 P05177 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8548608 0.88 MAPT (0.44) KMT2AMEN1TDP1ALDH1A1MAPT
SCHEMBL8551326 0.81 ALDH1A1 (0.44) KMT2AMEN1TDP1ALDH1A1MAPT
SCHEMBL8548327 0.77 ALDH1A1 (0.43) KMT2AALDH1A1MAPTLMNANPSR1
Hydrochloric Acid SCHEMBL8550917 0.76 PLAU (0.45) KMT2AMEN1TDP1ALDH1A1MAPT
SCHEMBL8550823 0.75 ALDH1A1 (0.42) KMT2AMEN1ALDH1A1MAPTLMNA
SCHEMBL8550890 0.74 ATM (0.55) KMT2AMEN1TDP1ALDH1A1MAPT
SCHEMBL8549262 0.74 ALDH1A1 (0.41) KMT2AMEN1ALDH1A1MAPTLMNA
SCHEMBL8552241 0.74 ALDH1A1 (0.41) KMT2AMEN1ALDH1A1MAPTLMNA
Hydrochloric Acid SCHEMBL8550910 0.74 ABCG2 (0.39) KMT2AMEN1TDP1ALDH1A1MAPT
SCHEMBL8548603 0.71 ALDH1A1 (0.50) KMT2AMEN1TDP1ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0825187-A1 Condensed pyridazinyl guanidines, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-02-25 EP disclosed