SCHEMBL8548917

SCHEMBL8548917

NS(=O)(=O)c1ccc(-c2onc(CC(=O)O)c2-c2ccc(Cl)cc2)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA P21397 2/20 0.45
MAOB P27338 2/20 0.45
CA1 P00915 9/20 0.43
CA2 P00918 9/20 0.43
CA4 P22748 6/20 0.43
CA7 P43166 4/20 0.43
PTGS2 P35354 7/20 0.43
CA9 Q16790 7/20 0.43
CA12 O43570 5/20 0.43
CA3 P07451 2/20 0.43
CA6 P23280 2/20 0.43
CA5A P35218 2/20 0.43
CA13 Q8N1Q1 2/20 0.43
CA14 Q9ULX7 2/20 0.43
CA5B Q9Y2D0 2/20 0.43
PTGS1 P23219 3/20 0.42
CHRNA7 P36544 1/20 0.42
S1PR1 P21453 1/20 0.40
MT-CO2 P00403 1/20 0.40
LMNA P02545 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6169911 0.90 PTGS2 (0.53) MAOAMAOBCA1CA2CA4
SCHEMBL8551541 0.87 PTGS2 (0.48) CA1CA2PTGS2CA9CA12
SCHEMBL6169927 0.79 PTGS2 (0.45) MAOAMAOBCA1CA2CA4
SCHEMBL6169873 0.79 PTGS2 (0.51) MAOAMAOBCA1CA2CA4
SCHEMBL6170883 0.79 PTGS2 (0.51) MAOAMAOBCA1CA2CA4
SCHEMBL5822486 0.78 PTGS2 (0.54) PTGS2PTGS1
SCHEMBL8593289 0.78 PTGS2 (0.51) PTGS2PTGS1
SCHEMBL6167881 0.78 PTGS2 (0.62) MAOAMAOBCA1CA2CA4
SCHEMBL6170394 0.77 CA1 (0.54) MAOAMAOBCA1CA2CA4
SCHEMBL6170551 0.77 CA1 (0.54) MAOAMAOBCA1CA2CA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0825989-A1 SUBSTITUTED OXAZOLES FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1998-03-04 EP disclosed