SCHEMBL8593289

SCHEMBL8593289

COc1ccc(-c2onc(CC(=O)O)c2-c2ccc(S(N)(=O)=O)cc2)cc1F

nearest known ligand 0.51

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 19/20 0.51
PTGS1 P23219 14/20 0.51
CDK2 P24941 1/20 0.44
ABCB11 O95342 1/20 0.43
ALDH1A1 P00352 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5822486 0.96 PTGS2 (0.54) PTGS2PTGS1CDK2ABCB11ALDH1A1
SCHEMBL6169532 0.88 PTGS2 (0.55) PTGS2PTGS1CDK2ABCB11ALDH1A1
SCHEMBL8551541 0.83 PTGS2 (0.48) PTGS2PTGS1
SCHEMBL6169911 0.80 PTGS2 (0.53) PTGS2PTGS1
SCHEMBL5732493 0.78 PTGS2 (0.51) PTGS2PTGS1CDK2ABCB11ALDH1A1
SCHEMBL5698527 0.78 PTGS2 (0.57) PTGS2PTGS1
SCHEMBL8548917 0.78 MAOA (0.45) PTGS2PTGS1
SCHEMBL4888033 0.77 PTGS2 (0.53) PTGS2PTGS1CDK2
SCHEMBL6168610 0.77 PTGS2 (0.51) PTGS2PTGS1
SCHEMBL6170005 0.76 PTGS2 (0.50) PTGS2PTGS1CDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0825989-A1 SUBSTITUTED OXAZOLES FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1998-03-04 EP disclosed