SCHEMBL8548976

SCHEMBL8548976

COc1ccc2c(c1OC)CC(NCC(O)c1cccc(C(F)(F)F)c1)C2

nearest known ligand 0.51

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ADRB3 P13945 2/20 0.42
NPC1 O15118 1/20 0.41
TP53 P04637 1/20 0.41
MAPT P10636 1/20 0.41
TSHR P16473 1/20 0.41
NFKB1 P19838 1/20 0.41
RAB9A P51151 1/20 0.41
NFKB2 Q00653 1/20 0.41
RELA Q04206 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
PNMT P11086 1/20 0.40
GRIN2B Q13224 3/20 0.40
ADRB1 P08588 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8546836 0.85 ADRB3 (0.56) ADRB3ADRB1
SCHEMBL8542977 0.73 ADRB3 (0.39) ADRB3GRIN2BADRB1
SCHEMBL8540992 0.72 AGTR2 (0.44) ADRB3ADRB1
SCHEMBL9241816 0.68 PNMT (0.46) TSHRNFKB1PNMTADRB1
SCHEMBL11339022 0.68 PNMT (0.46) TSHRNFKB1PNMTADRB1
SCHEMBL178870 0.68 MEN1 (0.55) MAPT
SCHEMBL178869 0.68 MEN1 (0.55) MAPT
SCHEMBL7148443 0.67 SMN1; SMN2 (0.50) ADRB3MAPTSMN1; SMN2ADRB1
SCHEMBL10974609 0.67 SMN1; SMN2 (0.50) ADRB3MAPTSMN1; SMN2ADRB1
SCHEMBL11288086 0.67 PNMT (0.44) PNMTGRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0608568-B1 Aminocycloalkanobenzodioxoles as beta-3 selective adrenergic agents AMERICAN CYANAMID CO (US) 1998-03-11 EP disclosed
US-5594027-A TREATMENT OF DIABETES, HYPERGLYCEMIA AND OBESITY AMERICAN CYANAMID COMPANY (US) 1997-01-14 US disclosed
US-5510376-A TREATING DIABETES, HYPERGLYCEMIA, OBESITY AMERICAN CYANAMID COMPANY (US) 1996-04-23 US disclosed
EP-0608568-A1 Aminocycloalkanobenzodioxoles as beta-3 selective adrenergic agents AMERICAN CYANAMID COMPANY (US) 1994-08-03 EP disclosed