SCHEMBL8540992

SCHEMBL8540992

COc1cccc(C(O)CNC2Cc3ccc(OCc4ccccc4)c(OCc4ccccc4)c3C2)c1

nearest known ligand 0.55

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
AGTR2 P50052 10/20 0.44
AGTR1 P30556 2/20 0.43
AOC3 Q16853 1/20 0.43
ADRB3 P13945 3/20 0.42
ADRB1 P08588 2/20 0.41
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
ACHE P22303 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8593552 0.91 ADRB3 (0.45) AGTR2ADRB3ADRB1
SCHEMBL9410787 0.79 AGTR2 (0.44) AGTR2AGTR1
SCHEMBL8549721 0.79 AGTR2 (0.44) AGTR2AGTR1AOC3
SCHEMBL8546836 0.74 ADRB3 (0.56) ADRB3ADRB1
SCHEMBL8978466 0.74 AGTR2 (0.44) AGTR2AGTR1CA1CA2ACHE
SCHEMBL8545450 0.74 AGTR2 (0.40) AGTR2AGTR1AOC3
SCHEMBL8548976 0.72 ADRB3 (0.42) ADRB3ADRB1
SCHEMBL8547546 0.71 CA1 (0.46) AGTR2AGTR1CA1CA2ACHE
SCHEMBL115985 0.71 ABCB1 (0.56) AOC3
SCHEMBL5142061 0.71 ADRB3 (0.49) ADRB3ADRB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0608568-B1 Aminocycloalkanobenzodioxoles as beta-3 selective adrenergic agents AMERICAN CYANAMID CO (US) 1998-03-11 EP disclosed
US-5594027-A TREATMENT OF DIABETES, HYPERGLYCEMIA AND OBESITY AMERICAN CYANAMID COMPANY (US) 1997-01-14 US disclosed
US-5510376-A TREATING DIABETES, HYPERGLYCEMIA, OBESITY AMERICAN CYANAMID COMPANY (US) 1996-04-23 US disclosed