SCHEMBL8549267

SCHEMBL8549267

CCCCCN1CCC(c2coc3ccc(NC(=O)Nc4cccc(C(=O)OC)c4)cc23)CC1

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 14/20 0.46
HTR2A P28223 13/20 0.46
DRD3 P35462 13/20 0.46
SLC6A4 P31645 1/20 0.45
NPC1 O15118 2/20 0.42
MAPT P10636 2/20 0.42
RAB9A P51151 2/20 0.42
ALDH1A1 P00352 1/20 0.42
CXCR3 P49682 1/20 0.41
MEN1 O00255 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
KMT2A Q03164 1/20 0.41
HTR7 P34969 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8548622 0.91 DRD2 (0.47) DRD2HTR2ADRD3SLC6A4
SCHEMBL8551604 0.89 UBE2M (0.49) DRD2HTR2ADRD3SLC6A4MAPT
SCHEMBL8703719 0.89 DRD2 (0.53) DRD2HTR2ADRD3SLC6A4
SCHEMBL8707882 0.86 DRD2 (0.54) DRD2HTR2ADRD3SLC6A4
SCHEMBL8551530 0.84 DRD2 (0.54) DRD2HTR2ADRD3SLC6A4
SCHEMBL7484342 0.84 HTR1D (0.58) DRD2
SCHEMBL8550671 0.83 DRD2 (0.56) DRD2HTR2ADRD3
SCHEMBL8703395 0.82 DRD2 (0.61) DRD2HTR2ADRD3SLC6A4
SCHEMBL8552841 0.82 KMT2A (0.47) DRD2HTR2ADRD3SLC6A4NPC1
SCHEMBL8703762 0.82 DRD2 (0.47) DRD2HTR2ADRD3SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5792763-A MIGRAINES; ANALGESICS; DISEASES LINKED TO DECREASED NEUROTRANMISSION OF SEROTONIN IN MAMMALS ELI LILLY AND COMPANY (US) 1998-08-11 US disclosed
EP-0835869-A2 New serotonin 5-HT1F agonists ELI LILLY AND COMPANY (US) 1998-04-15 EP disclosed