SCHEMBL8551730

SCHEMBL8551730

CN(C)CCCc1cc(N)cc2c1OCC2

nearest known ligand 0.35

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
NOS1 P29475 4/20 0.34
NOS3 P29474 2/20 0.34
NOS2 P35228 2/20 0.34
HTR1D P28221 1/20 0.32
HTR2C P28335 1/20 0.32
PARP1 P09874 1/20 0.31
PTGS1 P23219 1/20 0.31
PTGS2 P35354 1/20 0.31
SLC6A4 P31645 5/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8550551 0.74 HTR1B (0.41) NOS1NOS3NOS2HTR1DHTR2C
SCHEMBL8551471 0.73 KCNH2 (0.35) PARP1
SCHEMBL8551468 0.73 KCNH2 (0.35) PARP1
SCHEMBL5158843 0.73 NOS1 (0.43) NOS1NOS3NOS2SLC6A4
SCHEMBL8549330 0.72 L3MBTL4 (0.45) PARP1PTGS1PTGS2
SCHEMBL7484709 0.69 PARP1 (0.39) PARP1PTGS1PTGS2
SCHEMBL5160883 0.68 NOS1 (0.42) NOS1NOS3NOS2SLC6A4
SCHEMBL736186 0.68 PARP1 (0.42) PARP1
SCHEMBL14875929 0.66 NOS1 (0.40) NOS1NOS3NOS2SLC6A4
SCHEMBL9050184 0.66 PARP1 (0.39) PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0736025-B1 DYHYDROBENZOFURANYL-BIPHENYL CARBOXAMIDES HAVING 5HT1D ANTAGONISTIC ACTIVITY SMITHKLINE BEECHAM PLC (GB) 1998-07-22 EP disclosed
US-5700818-A Dihydrobenzofuranyl-biphenyl carboxamides having 5HT1D antagonistic activity SMITHKLINE BEECHAM P.L.C. (GB) 1997-12-23 US disclosed
EP-0736025-A1 DYHYDROBENZOFURANYL-BIPHENYL CARBOXAMIDES HAVING 5HT 1D? ANTAGONISTIC ACTIVITY SMITHKLINE BEECHAM PLC (GB) 1996-10-09 EP disclosed
WO-1995017401-A1 DYHYDROBENZOFURANYL-BIPHENYL CARBOXAMIDES HAVING 5HT1D ANTAGONISTIC ACTIVITY SMITHKLINE BEECHAM PLC (GB) 1995-06-29 WO disclosed