SCHEMBL8549474

SCHEMBL8549474

COc1ccc(C(=O)CN2CCC[C@H]2C(=O)NC(=O)c2ccccc2)cc1

nearest known ligand 0.56

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CTSK P43235 6/20 0.56
ALDH1A1 P00352 4/20 0.46
OPRM1 P35372 1/20 0.46
OPRK1 P41145 1/20 0.46
CYP2C9 P11712 1/20 0.46
CYP2C19 P33261 1/20 0.46
HTT P42858 2/20 0.46
ALOX15 P16050 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
SCN5A Q14524 1/20 0.45
SCN2A Q99250 1/20 0.45
CHRM3 P20309 1/20 0.45
MAPK1 P28482 1/20 0.44
HPGD P15428 2/20 0.44
POLB P06746 1/20 0.44
DPP4 P27487 1/20 0.44
ALOX5 P09917 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8549483 1.00 CTSK (0.56) CTSKALDH1A1OPRM1OPRK1CYP2C9
SCHEMBL8544621 0.90 CTSK (0.47) CTSKALDH1A1OPRM1OPRK1HPGD
SCHEMBL8544615 0.90 CTSK (0.47) CTSKALDH1A1OPRM1OPRK1HPGD
SCHEMBL8543316 0.90 CTSK (0.53) CTSKALDH1A1HPGDDPP4
SCHEMBL8543314 0.90 CTSK (0.53) CTSKALDH1A1HPGDDPP4
SCHEMBL8548127 0.90 MEN1 (0.51) CTSKALDH1A1SMN1; SMN2MAPK1
SCHEMBL8548133 0.90 MEN1 (0.51) CTSKALDH1A1SMN1; SMN2MAPK1
SCHEMBL8548482 0.88 CTSK (0.46) CTSKALDH1A1SMN1; SMN2
SCHEMBL8548689 0.88 PTGER4 (0.49) CTSK
SCHEMBL8548691 0.88 PTGER4 (0.49) CTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0564924-B1 2-Oxoethyl derivatives as immunosuppressants BAYER AG (US) 1998-09-09 EP claimed
EP-0564924-A2 2-Oxoethyl derivatives as immunosuppressants Bayer Corporation (US) 1993-10-13 EP claimed
EP-0564924-B1 2-Oxoethyl derivatives as immunosuppressants BAYER AG (US) 1998-09-09 EP disclosed
US-5686424-A FOR TREATING INFLAMMATION MILES INC. (US) 1997-11-11 US disclosed
EP-0564924-A2 2-Oxoethyl derivatives as immunosuppressants Bayer Corporation (US) 1993-10-13 EP disclosed