SCHEMBL8549574

SCHEMBL8549574

CCOC(=O)Oc1c(-c2ccc(OC)cc2OCC(=O)O)c2cc(OC)c(OC3CCCC3)cc2n1Cc1ccc2nsnc2c1

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
EDNRB P24530 6/20 0.43
EDNRA P25101 2/20 0.43
PDE4B Q07343 5/20 0.37
PDE4D Q08499 4/20 0.37
PDE4A P27815 3/20 0.37
PDE4C Q08493 3/20 0.37
PTGDR2 Q9Y5Y4 1/20 0.33
KDM4E B2RXH2 1/20 0.33
GAA P10253 1/20 0.33
HSD17B10 Q99714 1/20 0.33
HTT P42858 2/20 0.32
ALDH1A1 P00352 1/20 0.32
ELANE P08246 1/20 0.32
KMT2A Q03164 2/20 0.32
MEN1 O00255 1/20 0.32
PTPN1 P18031 2/20 0.32
USP2 O75604 1/20 0.32
ALOX5AP P20292 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8550648 0.98 EDNRB (0.42) EDNRBEDNRAPDE4BPDE4DPDE4A
SCHEMBL8547930 0.93 EDNRB (0.47) EDNRBEDNRAKDM4EGAAHSD17B10
SCHEMBL8547478 0.88 EDNRB (0.43) EDNRBEDNRAKDM4EGAAHSD17B10
SCHEMBL8547163 0.88 EDNRB (0.45) EDNRBEDNRAKDM4EGAAHSD17B10
SCHEMBL8549318 0.88 EDNRB (0.43) EDNRBEDNRAKDM4EHTTPTPN1
SCHEMBL8547597 0.85 EDNRB (0.47) EDNRBEDNRAPDE4BPDE4DPDE4A
SCHEMBL8549234 0.85 EDNRB (0.52) EDNRBEDNRAPTGDR2KDM4EGAA
SCHEMBL8547864 0.85 EDNRB (0.49) EDNRBEDNRAPTPN1
SCHEMBL8546037 0.83 EDNRB (0.60) EDNRBEDNRAPTGDR2KDM4EGAA
SCHEMBL8547128 0.83 EDNRB (0.49) EDNRBEDNRAPDE4BPDE4DPDE4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0863898-A1 ENDOTHELIN RECEPTOR ANTAGONISTS MERCK PATENT GmbH (DE) 1998-09-16 EP disclosed
WO-1997019077-A1 ENDOTHELIN RECEPTOR ANTAGONISTS MERCK Patent Gesellschaft mit beschränkter Haftung (DE) 1997-05-29 WO disclosed