SCHEMBL8550210

SCHEMBL8550210

Nc1cc(Cl)ccc1C(=O)OC1CCN(Cc2ccccc2)CC1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A12 P48065 1/20 0.54
BCHE P06276 2/20 0.53
DRD2 P14416 2/20 0.50
DRD4 P21917 2/20 0.50
OPRK1 P41145 2/20 0.48
SIGMAR1 Q99720 3/20 0.47
KDM4E B2RXH2 2/20 0.47
ALDH1A1 P00352 2/20 0.47
ACHE P22303 2/20 0.47
CYP1A2 P05177 1/20 0.47
CYP3A4 P08684 1/20 0.47
ADRA2A P08913 1/20 0.47
CYP2D6 P10635 1/20 0.47
CYP2C9 P11712 1/20 0.47
ADRA2B P18089 1/20 0.47
ADRA2C P18825 1/20 0.47
SLC6A2 P23975 1/20 0.47
HTR2A P28223 1/20 0.47
HTR2C P28335 1/20 0.47
ADRA1A P35348 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8550148 0.99 SLC6A12 (0.53) SLC6A12BCHEDRD2DRD4OPRK1
SCHEMBL8553603 0.90 BCHE (0.54) SLC6A12BCHEDRD2DRD4OPRK1
SCHEMBL8552042 0.89 BCHE (0.53) SLC6A12BCHEOPRK1SIGMAR1
Hydrochloric Acid SCHEMBL8553924 0.89 BCHE (0.53) SLC6A12BCHEDRD2DRD4OPRK1
SCHEMBL8550767 0.88 BCHE (0.52) BCHEDRD2DRD4OPRK1ACHE
SCHEMBL8551172 0.88 BCHE (0.52) BCHEDRD2DRD4OPRK1SIGMAR1
SCHEMBL8551366 0.88 BCHE (0.52) BCHEDRD2DRD4OPRK1SIGMAR1
Hydrochloric Acid SCHEMBL8554134 0.88 BCHE (0.52) SLC6A12BCHEOPRK1SIGMAR1
SCHEMBL8551180 0.87 BCHE (0.58) BCHEOPRK1SIGMAR1KDM4EALDH1A1
Hydrochloric Acid SCHEMBL8554127 0.87 BCHE (0.51) BCHEDRD2DRD4OPRK1SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1084329-C Benzyl piepridine derivs as pharmaceutical agents HOFFMANN LA ROCHE (CH) 2002-05-08 CN disclosed
EP-0871613-A1 BENZYL PIPERIDINE DERIVATIVES AS PHARMACEUTICAL AGENTS F. HOFFMANN-LA ROCHE AG (CH) 1998-10-21 EP disclosed
CN-1183768-A Benzyl piepridine derivs as pharmaceutical agents HOFFMANN LA ROCHE (CH) 1998-06-03 CN disclosed
US-5753679-A SCIZOPHRENIA HOFFMANN-LA ROCHE INC. (US) 1998-05-19 US disclosed
WO-1996035666-A1 BENZYL PIPERIDINE DERIVATIVES AS PHARMACEUTICAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 1996-11-14 WO disclosed